TCS-OX2-29
CAS No. 372523-75-6
TCS-OX2-29 ( —— )
Catalog No. M19326 CAS No. 372523-75-6
TCS-OX2-29 is a potent and selective OX2 receptor antagonist (IC50: 40 nM). It displays >250-fold selectivity for OX2 over OX1.
Purity : 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
2MG | 35 | In Stock |
|
5MG | 58 | In Stock |
|
10MG | 87 | In Stock |
|
25MG | 170 | In Stock |
|
50MG | 250 | In Stock |
|
100MG | 447 | In Stock |
|
200MG | Get Quote | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
|
Biological Information
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Product NameTCS-OX2-29
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NoteResearch use only, not for human use.
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Brief DescriptionTCS-OX2-29 is a potent and selective OX2 receptor antagonist (IC50: 40 nM). It displays >250-fold selectivity for OX2 over OX1.
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DescriptionTCS-OX2-29 is a potent and selective OX2 receptor antagonist (IC50: 40 nM). It displays >250-fold selectivity for OX2 over OX1.
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Synonyms——
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PathwayCytoskeleton/Cell Adhesion Molecules
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TargetKinesin
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RecptorOX2
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number372523-75-6
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Formula Weight397.51
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Molecular FormulaC23H31N3O3
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Purity98%
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SolubilityH2O : < 0.1 mg/mL
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SMILESCOC1=C(OC)C=C2CN(CCC2=C1)C(=O)[C@@H](NCC1=CC=NC=C1)C(C)(C)C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Hirose M et al. N-acyl 6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline: the first orexin-2 receptor selective non-peptidicantagonist. Bioorg Med Chem Lett, 2003 Dec 15, 13(24):4497-9.
molnova catalog
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