Paprotrain

CAS No. 57046-73-8

Paprotrain ( (alphaZ)-alpha-(3-Pyridinylmethylene)-1H-indole-3-acetonitrile )

Catalog No. M26357 CAS No. 57046-73-8

Paprotrain inhibits the ATPase activity of MKLP-2 with an IC50 of 1.35 μM and a Ki of 3.36 μM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 42 Get Quote
10MG 60 Get Quote
25MG 105 Get Quote
50MG 168 Get Quote
100MG 303 Get Quote
200MG 443 Get Quote
500MG 707 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    Paprotrain
  • Note
    Research use only, not for human use.
  • Brief Description
    Paprotrain inhibits the ATPase activity of MKLP-2 with an IC50 of 1.35 μM and a Ki of 3.36 μM.
  • Description
    Paprotrain inhibits the ATPase activity of MKLP-2 with an IC50 of 1.35 μM and a Ki of 3.36 μM.(In Vitro):Paprotrain-treated porcine oocytes suffer failure of nuclear maturation.?The number of oocytes arrested at early MI stage increase in a dose-dependent manner after KIF20A activity inhibition, while the percentage of oocytes that reach ATI and MII stages decrease after treatment.
  • Synonyms
    (alphaZ)-alpha-(3-Pyridinylmethylene)-1H-indole-3-acetonitrile
  • Pathway
    Cytoskeleton/Cell Adhesion Molecules
  • Target
    Kinesin
  • Recptor
    ——
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    57046-73-8
  • Formula Weight
    245.3
  • Molecular Formula
    C16H11N3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    N#C\C(=C/c1cccnc1)c1c[nH]c2ccccc12
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Kennedy GL Jr, Chen HC, Hall GT. Inhalation toxicity of dehydrothio-p-toluidine. Food Chem Toxicol. 1984 Apr;22(4):289-92.
molnova catalog
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