JAK3/BTK-IN-1

CAS No. 2674036-91-8

JAK3/BTK-IN-1( —— )

Catalog No. M37669 CAS No. 2674036-91-8

JAK3/ BTk-in-1 is a dual JAK3/BTK inhibitor that specifically targets and inhibits Janus kinase 3 (JAK3) and Bruton's tyrosine kinase (BTK), two important targets in autoimmune diseases.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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25MG 1264 In Stock
50MG 1600 In Stock
100MG 2409 In Stock
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Biological Information

  • Product Name
    JAK3/BTK-IN-1
  • Note
    Research use only, not for human use.
  • Brief Description
    JAK3/ BTk-in-1 is a dual JAK3/BTK inhibitor that specifically targets and inhibits Janus kinase 3 (JAK3) and Bruton's tyrosine kinase (BTK), two important targets in autoimmune diseases.
  • Description
    JAK3/BTK-IN-1 is a potent inhibitor of JAK3/BTK. BTK and JAK3 are two important targets for autoimmune diseases. Simultaneous inhibition of the BTK/JAK3 signalling pathway exhibits synergistic effects. JAK3/BTK-IN-1 has the potential for the research of JAK3 kinase and/or BTK-related diseases (extracted from patent WO2021147952A1, compound 002).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Tyrosine Kinase
  • Target
    BTK
  • Recptor
    BTK | JAK
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2674036-91-8
  • Formula Weight
    456.54
  • Molecular Formula
    C25H28N8O
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    N(C1=C2C(=CNC2=NC(NC3=CN(CC)N=C3)=N1)C4=CC=CC=C4)[C@H]5CN(C(C=C)=O)CCC5
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Guobao Zhang, et al. Pyrimidopyrroles. Patent WO2021147952A1.
molnova catalog
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