Tiapamil hydrochloride

CAS No. 57010-32-9

Tiapamil hydrochloride( —— )

Catalog No. M33148 CAS No. 57010-32-9

Tiapamil hydrochloride (Ro 11-1781 hydrochloride) is a calcium channel blocker with antihypertensive activity and may be used in the study of angina and cardiovascular disease.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 414 In Stock
5MG 686 In Stock
10MG 938 In Stock
25MG 1444 In Stock
50MG 1841 In Stock
100MG Get Quote In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Tiapamil hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    Tiapamil hydrochloride (Ro 11-1781 hydrochloride) is a calcium channel blocker with antihypertensive activity and may be used in the study of angina and cardiovascular disease.
  • Description
    Tiapamil hydrochloride is a calcium channel blocker.
  • In Vitro
    Tiapamil, a new calcium antagonist: hemodynamic effects in patients with acute myocardial infarction. Tiapamil is a new verapamil congener.Without precipitating left ventricular failure, Tiapamil reduced afterload and heart rate and maintained cardiac index while apparently improving diastolic compliance. Tiapamil, a new calcium channel blocking agent with anti-anginal efficacy.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Calcium Channel
  • Recptor
    Calcium Channel
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    57010-32-9
  • Formula Weight
    592.16
  • Molecular Formula
    C26H38ClNO8S2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    Cl.O=S1(=O)CCCS(=O)(=O)C1(C2=CC=C(OC)C(OC)=C2)CCCN(C)CCC3=CC=C(OC)C(OC)=C3
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Eichler HG, et al. Tiapamil, a new calcium antagonist: hemodynamic effects in patients with acute myocardial infarction. Circulation. 1985 Apr;71(4):779-86.?
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