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PROTAC BRD4 ligand-1
CAS No. 2313230-51-0
PROTAC BRD4 ligand-1( —— )
Catalog No. M33078 CAS No. 2313230-51-0
PROTAC BRD4 ligand-1, a component of Protac GNE-987, is a ligand for BRD4 and acts as an inhibitor of BET.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 297 | In Stock |
|
| 10MG | 496 | In Stock |
|
| 25MG | 938 | In Stock |
|
| 50MG | 1544 | In Stock |
|
| 100MG | 2223 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePROTAC BRD4 ligand-1
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NoteResearch use only, not for human use.
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Brief DescriptionPROTAC BRD4 ligand-1, a component of Protac GNE-987, is a ligand for BRD4 and acts as an inhibitor of BET.
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DescriptionPROTAC BRD4 ligand-1 is a potent BET inhibitor and a ligand for target BRD4 protein for PROTACT GNE-987 (HY-129937A).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayChromatin/Epigenetic
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TargetEpigenetic Reader Domain
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RecptorEpigenetic Reader Domain | Ligands for Target Protein for PROTAC
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Research Area——
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Indication——
Chemical Information
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CAS Number2313230-51-0
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Formula Weight500.47
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Molecular FormulaC23H18F2N4O5S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 5 mg/mL (9.99 mM; Ultrasonic )
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SMILESCn1cc2-c3cc(CS(C)(=O)=O)c(cc3N(Cc3c[nH]c(c23)c1=O)c1ncc(F)cc1F)C(O)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Pillow TH, et al. Antibody Conjugation of a Chimeric BET Degrader Enables in vivo Activity. ChemMedChem. 2019 Oct 31.?
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