BD 1008 dihydrobromide

CAS No. 138356-09-9

BD 1008 dihydrobromide( —— )

Catalog No. M27463 CAS No. 138356-09-9

BD1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 284 Get Quote
10MG 444 Get Quote
25MG 647 Get Quote
50MG 851 Get Quote
100MG 1269 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    BD 1008 dihydrobromide
  • Note
    Research use only, not for human use.
  • Brief Description
    BD1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM).
  • Description
    BD1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM). BD1008 dihydrobromide have high affinity for sigma1 receptors, moderate affinity for sigma2 receptors. BD1008 dihydrobromide attenuate the toxicity and stimulant effects of cocaine through antagonism of sigma receptors.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Autophagy
  • Target
    Sigma receptor
  • Recptor
    ——
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    138356-09-9
  • Formula Weight
    463.08
  • Molecular Formula
    C15H24Br2Cl2N2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    Br.Br.CN(CCN1CCCC1)CCc1ccc(Cl)c(Cl)c1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Barakat MT, et al. Simethicone is retained in endoscopes despite reprocessing: impact of its use on working channel fluid retention and adenosine triphosphate bioluminescence values (with video). Gastrointest Endosc. 2018 Aug 17.
molnova catalog
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