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BD 1008 dihydrobromide
CAS No. 138356-09-9
BD 1008 dihydrobromide( —— )
Catalog No. M27463 CAS No. 138356-09-9
BD1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 69 | In Stock |
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| 2MG | 33 | In Stock |
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| 5MG | 53 | In Stock |
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| 10MG | 93 | In Stock |
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| 25MG | 227 | In Stock |
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| 50MG | 347 | In Stock |
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| 100MG | 494 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBD 1008 dihydrobromide
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NoteResearch use only, not for human use.
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Brief DescriptionBD1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM).
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DescriptionBD1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM). BD1008 dihydrobromide have high affinity for sigma1 receptors, moderate affinity for sigma2 receptors. BD1008 dihydrobromide attenuate the toxicity and stimulant effects of cocaine through antagonism of sigma receptors.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayAutophagy
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TargetSigma receptor
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number138356-09-9
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Formula Weight463.08
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Molecular FormulaC15H24Br2Cl2N2
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Purity>98% (HPLC)
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Solubility——
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SMILESBr.Br.CN(CCN1CCCC1)CCc1ccc(Cl)c(Cl)c1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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4-PPBP maleate
4-PPBP maleate is a potent σ1 receptor (ligand) agonist and a selective, non-competitive NR1a/2B NMDA receptor antagonist in the context of Xenopus oocytes expression, with neuroprotective properties.
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PD 144418 oxalate
PD 144418 oxalate is a highly potent and selective sigma 1 (σ1) receptor ligand with a Ki value of 0.08 nM for σ1 and 1377 nM for σ2, exhibiting negligible affinity for other receptors, ion channels, and enzymes, and demonstrating potential antipsychotic activity.
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KB-5492 free base
KB-5492 free base is an orally available and selective antiulcer agent that inhibits sigma receptors, inhibits [3H]1,3-di(2-tolyl)guanidine (DTG) binding to sigma receptors, and may be useful in the study of gastric lesions and gastric secretion.
