ODM-207

CAS No. 1801503-93-4

ODM-207( BET-IN-4 | ODM-207 | ODM207 )

Catalog No. M26070 CAS No. 1801503-93-4

BET-IN-4 is a potent BRD4 inhibitor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 86 Get Quote
5MG 132 Get Quote
10MG 215 Get Quote
25MG 393 Get Quote
50MG 565 Get Quote
100MG 800 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    ODM-207
  • Note
    Research use only, not for human use.
  • Brief Description
    BET-IN-4 is a potent BRD4 inhibitor.
  • Description
    BET-IN-4 is a potent BRD4 inhibitor.(In Vitro):BET-IN-4 inhibits BRD4 with an IC50 of ≤ 1 μM.
  • In Vitro
    ODM-207 (Compound 50) is a potent BET bromodomain protein (BRD4) inhibitor, with an IC50 of ≤ 1 μM.
  • In Vivo
    ——
  • Synonyms
    BET-IN-4 | ODM-207 | ODM207
  • Pathway
    Chromatin/Epigenetic
  • Target
    Epigenetic Reader Domain
  • Recptor
    ——
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1801503-93-4
  • Formula Weight
    375.428
  • Molecular Formula
    C22H21N3O3
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 10 mg/mL (26.64 mM)
  • SMILES
    COc1cc2n(Cc3ccccn3)c(=O)c(C)cc2cc1-c1c(C)noc1C
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Kao-Lu Pan, et al. Identification of trans,trans-2,4-decadienal metabolites in mouse and human cells using liquid chromatography-mass spectrometry. Chem Res Toxicol. 2014 Oct 20;27(10):1707-19.
molnova catalog
related products
  • IRAK4-IN-1

    IRAK4-IN-1 is an interleukin-1 receptor associated kinase 4 (IRAK4) inhibitor with an IC50 of 7 nM.

  • Y06137

    Y06137 is an effective and selective BET inhibitor with a Kd of 81 nM for BRD4(1) bromodomain. Y06137 can be used for research on the treatment of castration-resistant prostate cancer.

  • CTB

    CTB (Cholera Toxin B subunit) is an activator of p300 histone acetyltransferase and induces apoptosis in MCF-7 cells.