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ODM-207
CAS No. 1801503-93-4
ODM-207( BET-IN-4 | ODM-207 | ODM207 )
Catalog No. M26070 CAS No. 1801503-93-4
BET-IN-4 is a potent BRD4 inhibitor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 92 | In Stock |
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| 5MG | 84 | In Stock |
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| 10MG | 136 | In Stock |
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| 25MG | 249 | In Stock |
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| 50MG | 351 | In Stock |
|
| 100MG | 496 | In Stock |
|
| 200MG | 682 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameODM-207
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NoteResearch use only, not for human use.
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Brief DescriptionBET-IN-4 is a potent BRD4 inhibitor.
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DescriptionBET-IN-4 is a potent BRD4 inhibitor.(In Vitro):BET-IN-4 inhibits BRD4 with an IC50 of ≤ 1 μM.
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In VitroODM-207 (Compound 50) is a potent BET bromodomain protein (BRD4) inhibitor, with an IC50 of ≤ 1 μM.
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In Vivo——
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SynonymsBET-IN-4 | ODM-207 | ODM207
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PathwayChromatin/Epigenetic
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TargetEpigenetic Reader Domain
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number1801503-93-4
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Formula Weight375.428
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Molecular FormulaC22H21N3O3
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 10 mg/mL (26.64 mM)
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SMILESCOc1cc2n(Cc3ccccn3)c(=O)c(C)cc2cc1-c1c(C)noc1C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Kao-Lu Pan, et al. Identification of trans,trans-2,4-decadienal metabolites in mouse and human cells using liquid chromatography-mass spectrometry. Chem Res Toxicol. 2014 Oct 20;27(10):1707-19.
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