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RBN012759
CAS No. 2360851-29-0
RBN012759( —— )
Catalog No. M22469 CAS No. 2360851-29-0
RBN012759, a potent and selective PARP14 inhibitor, decreases pro-tumor macrophage function and elicits inflammatory responses in tumor explants.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 274 | In Stock |
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| 2MG | 149 | In Stock |
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| 5MG | 250 | In Stock |
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| 10MG | 372 | In Stock |
|
| 25MG | 645 | In Stock |
|
| 50MG | 918 | In Stock |
|
| 100MG | 1283 | In Stock |
|
| 200MG | 1730 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameRBN012759
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NoteResearch use only, not for human use.
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Brief DescriptionRBN012759, a potent and selective PARP14 inhibitor, decreases pro-tumor macrophage function and elicits inflammatory responses in tumor explants.
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DescriptionRBN012759, a potent and selective PARP14 inhibitor, decreases pro-tumor macrophage function and elicits inflammatory responses in tumor explants.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayCell Cycle/DNA Damage
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TargetPARP
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RecptorPARP14
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Research Area——
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Indication——
Chemical Information
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CAS Number2360851-29-0
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Formula Weight378.46
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Molecular FormulaC19H23FN2O3S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 250 mg/mL (660.57 mM)
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SMILESO[C@H]1CC[C@@H](CC1)SCc1nc2cc(OCC3CC3)cc(F)c2c(=O)[nH]1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Schenkel L, et, al. A potent and selective PARP14 inhibitor decreases pro-tumor macrophage function and elicits inflammatory responses in tumor explants. AACR Annual Meeting 2020.
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