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BYK204165

CAS No. 1104546-89-5

BYK204165( RT-017290 )

Catalog No. M21123 CAS No. 1104546-89-5

BYK204165 is a potent PARP inhibitor (PARP1; IC50 = 44.67 nM for human recombinant PARP1 in an enzyme assay).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 67 In Stock
5MG 61 In Stock
10MG 92 In Stock
25MG 170 In Stock
50MG 245 In Stock
100MG 361 In Stock
200MG 528 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock
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Biological Information

  • Product Name
    BYK204165
  • Note
    Research use only, not for human use.
  • Brief Description
    BYK204165 is a potent PARP inhibitor (PARP1; IC50 = 44.67 nM for human recombinant PARP1 in an enzyme assay).
  • Description
    BYK204165 is a potent PARP inhibitor (PARP1; IC50 = 44.67 nM for human recombinant PARP1 in an enzyme assay).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    RT-017290
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    PARP
  • Recptor
    PARP
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1104546-89-5
  • Formula Weight
    252
  • Molecular Formula
    C15H12N2O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:125 mg/mL (495.50 mM; Need ultrasonic)
  • SMILES
    Cn1cccc1C=C1C(=O)NC(=O)c2ccccc21
  • Chemical Name
    (4Z)-4-[(1-methylpyrrol-2-yl)methylidene]isoquinoline-13-dione

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Eltze T Boer R Wagner T et al. Imidazoquinolinone imidazopyridine and isoquinolindione derivatives as novel and potent inhibitors of the poly(ADP-ribose) polymerase (PARP): a comparison with standard PARP inhibitors.[J]. molecular pharmacology 2008 74(6):1587-1598.
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