GW 405833

CAS No. 180002-83-9

GW 405833( L-768242 )

Catalog No. M20934 CAS No. 180002-83-9

GW 405833 is an agonist of cannabinoid-2 (CB(2)) receptor-selective.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 75 In Stock
5MG 76 In Stock
10MG 116 In Stock
25MG 211 In Stock
50MG 323 In Stock
100MG 479 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    GW 405833
  • Note
    Research use only, not for human use.
  • Brief Description
    GW 405833 is an agonist of cannabinoid-2 (CB(2)) receptor-selective.
  • Description
    GW 405833 is an agonist of cannabinoid-2 (CB(2)) receptor-selective.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    L-768242
  • Pathway
    GPCR/G Protein
  • Target
    Cannabinoid Receptor
  • Recptor
    CB2
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    180002-83-9
  • Formula Weight
    447.35
  • Molecular Formula
    C23H24Cl2N2O3
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 125 mg/mL (279.42 mM)
  • SMILES
    COc1ccc2c(c1)c(CCN1CCOCC1)c(C)n2C(=O)c1cccc(Cl)c1Cl
  • Chemical Name
    1-(23-Dichlorobenzoyl)-5-methoxy-2-methyl-3-(2-morpholinoethyl)-1H-indole

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Li A L Carey L M Mackie K et al. The cannabinoid CB 2 agonist GW405833 suppresses inflammatory and neuropathic pain through a CB 1 mechanism that is independent of CB 2 receptors in mice[J]. Journal of Pharmacology and Experimental Therapeutics 2017 362(2):jpet.117.241901.
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