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GAT-211

CAS No. 102704-40-5

GAT-211( GAT211 )

Catalog No. M10132 CAS No. 102704-40-5

GAT-211 (GAT211) is a selective cannabinoid 1 receptor (CB1R) positive allosteric modulator with pKb of 7.26, Arrestin2 EC50 of 775 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 67 In Stock
5MG 61 In Stock
10MG 92 In Stock
25MG 151 In Stock
50MG 217 In Stock
100MG 321 In Stock
200MG Get Quote In Stock
500MG 775 In Stock
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Biological Information

  • Product Name
    GAT-211
  • Note
    Research use only, not for human use.
  • Brief Description
    GAT-211 (GAT211) is a selective cannabinoid 1 receptor (CB1R) positive allosteric modulator with pKb of 7.26, Arrestin2 EC50 of 775 nM.
  • Description
    GAT-211 (GAT211) is a selective cannabinoid 1 receptor (CB1R) positive allosteric modulator with pKb of 7.26, Arrestin2 EC50 of 775 nM; engages CB1R allosteric site(s), enhances the binding of the orthosteric full agonist [3H]CP55,490, and reduces the binding of the orthosteric antagonist/inverse agonist [3H]SR141716A; displayed both PAM and agonist activity in HEK293A and Neuro2a cells expressing human recombinant CB1R (hCB1R) and in mouse-brain membranes rich in native CB1R.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    GAT211
  • Pathway
    GPCR/G Protein
  • Target
    Cannabinoid Receptor
  • Recptor
    Cannabinoid Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    102704-40-5
  • Formula Weight
    342.4
  • Molecular Formula
    C22H18N2O2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (292.06 mM)
  • SMILES
    O=[N+](CC(C1=C(C2=CC=CC=C2)NC3=C1C=CC=C3)C4=CC=CC=C4)[O-]
  • Chemical Name
    3-(2-nitro-1-phenylethyl)-2-phenyl-1H-indole

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Laprairie RB, et al. ACS Chem Neurosci. 2017 Jun 21;8(6):1188-1203.
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