Triprolidine hydrochloride

CAS No. 6138-79-0

Triprolidine hydrochloride( —— )

Catalog No. M15313 CAS No. 6138-79-0

Histamine H1 antagonist used in allergic rhinitis; asthma; and urticaria.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 32 In Stock
10MG 29 In Stock
25MG 61 In Stock
50MG 90 In Stock
100MG 133 In Stock
200MG Get Quote In Stock
500MG 331 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Triprolidine hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    Histamine H1 antagonist used in allergic rhinitis; asthma; and urticaria.
  • Description
    Histamine H1 antagonist used in allergic rhinitis; asthma; and urticaria. It is a component of COUGH and COLD medicines. It may cause drowsiness.(In Vivo):Triprolidine hydrochloride monohydrate (292.81-1467.20 μg/kg; intrathecal injection) produces a dose-dependent effect of spinal motor and sensory block in rats.
  • In Vitro
    ——
  • In Vivo
    Triprolidine hydrochloride monohydrate (292.81-1467.20 μg/kg; intrathecal injection) produces a dose-dependent effect of spinal motor and sensory block in rats. Animal Model:Male Sprague-Dawley rat (300-350 g)Dosage:292.81 μg/kg, 488.02 μg/kg, 733.60μg/kg, 1098.83 μg/kg, 1467.20 μg/kg Administration:Intrathecal injection Result:Elicited a dose-dependent spinal block.
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Histamine Receptor
  • Recptor
    H1 receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    6138-79-0
  • Formula Weight
    314.85
  • Molecular Formula
    C19H23ClN2
  • Purity
    >98% (HPLC)
  • Solubility
    Soluble in Water
  • SMILES
    CC1=CC=C(C=C1)/C(=C\CN2CCCC2)/C3=CC=CC=N3.Cl
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Hansen EB Jr, et al. J Pharm Sci. 1988 Mar;77(3):259-64.
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