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Astemizole
CAS No. 68844-77-9
Astemizole( NSC 329963 )
Catalog No. M15631 CAS No. 68844-77-9
Antihistamine drug now withdrawn from the market in many countries because of rare but potentially fatal side effects.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 44 | In Stock |
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| 5MG | 40 | In Stock |
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| 10MG | 55 | In Stock |
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| 25MG | 89 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameAstemizole
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NoteResearch use only, not for human use.
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Brief DescriptionAntihistamine drug now withdrawn from the market in many countries because of rare but potentially fatal side effects.
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DescriptionAntihistamine drug now withdrawn from the market in many countries because of rare but potentially fatal side effects.
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In Vitro——
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In Vivo——
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SynonymsNSC 329963
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PathwayGPCR/G Protein
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TargetHistamine Receptor
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RecptorH1 receptor| Potassium Channel
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Research AreaInflammation/Immunology
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Indication——
Chemical Information
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CAS Number68844-77-9
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Formula Weight458.58
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Molecular FormulaC28H31FN4O
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Purity>98% (HPLC)
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SolubilityWater: 432 mg/L
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SMILESCOC1=CC=C(C=C1)CCN2CCC(CC2)NC3=NC4=CC=CC=C4N3CC5=CC=C(C=C5)F
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Chemical Name1-[(4-fluorophenyl)methyl]-N-[1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl]benzimidazol-2-amine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Salata JJ, et al. Circ Res. 1995 Jan;76(1):110-9.
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