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GLUT4-IN-17
CAS No. 1061081-61-5
GLUT4-IN-17( —— )
Catalog No. M10271 CAS No. 1061081-61-5
A potent, selective glucose transporter 4 (GLUT4) inhibitor with IC450 of 10.8 uM, inhibits MM cell proliferation.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameGLUT4-IN-17
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NoteResearch use only, not for human use.
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Brief DescriptionA potent, selective glucose transporter 4 (GLUT4) inhibitor with IC450 of 10.8 uM, inhibits MM cell proliferation.
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DescriptionA potent, selective glucose transporter 4 (GLUT4) inhibitor with IC450 of 10.8 uM, inhibits MM cell proliferation; reduces ATB-BMPA binding to GLUT4 to a much greater extent than to GLUT1, inhibits 2-DOG uptake in GLUT4-expressing cells.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMembrane Transporter/Ion Channel
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TargetGLUT
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RecptorGLUT
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Research Area——
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Indication——
Chemical Information
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CAS Number1061081-61-5
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Formula Weight509.654
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Molecular FormulaC31H35N5O2
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name(3-((3-((methyl(quinolin-6-ylmethyl)amino)methyl)phenoxy)methyl)piperidin-1-yl)(1,4,5,6-tetrahydrocyclopenta[c]pyrazol-3-yl)methanone
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Mishra RK, et al. J Biol Chem. 2015 Jun 5;290(23):14441-53.
molnova catalog
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