CIM0216

CAS No. 1031496-06-6

CIM0216 ( N-(5-methyl-1,2-oxazol-3-yl)-2-phenyl-2-(1,2,3,4-tetrahydroquinolin-1-yl)acetamide )

Catalog No. M23235 CAS No. 1031496-06-6

CIM0216 is a synthetic TRPM3 activator whose potency and apparent affinity greatly exceeds that of the canonical TRPM3 agonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 49 In Stock
5MG 76 In Stock
10MG 133 In Stock
25MG 282 In Stock
50MG 441 In Stock
100MG 664 In Stock
500MG 1377 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    CIM0216
  • Note
    Research use only, not for human use.
  • Brief Description
    CIM0216 is a synthetic TRPM3 activator whose potency and apparent affinity greatly exceeds that of the canonical TRPM3 agonist.
  • Description
    CIM0216 is a synthetic TRPM3 activator whose potency and apparent affinity greatly exceeds that of the canonical TRPM3 agonist.
  • Synonyms
    N-(5-methyl-1,2-oxazol-3-yl)-2-phenyl-2-(1,2,3,4-tetrahydroquinolin-1-yl)acetamide
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    TRP/TRPV Channel
  • Recptor
    TRPM3
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1031496-06-6
  • Formula Weight
    347.4
  • Molecular Formula
    C21H21N3O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 30 mg/mL?(86.35 mM;?Need ultrasonic and warming);Ethanol: 17 mg/mL?(48.93 mM;?Need ultrasonic and warming)
  • SMILES
    O=C(NC1=NOC(C)=C1)C(C2=CC=CC=C2)N3CCCC4=C3C=CC=C4
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Vriens J , Owsianik G , Hofmann T , et al. TRPM3 is a nociceptor channel involved in the detection of noxious heat.[J]. Neuron, 2011, 70(3):482-494.
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