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BMS-986020
CAS No. 1257213-50-5
BMS-986020 ( BMS 986020;BMS986020;AM-152;AM152;AM 152 )
Catalog No. M11058 CAS No. 1257213-50-5
BMS-986020 (BMS986020, AM-152) is a potent, selective, orally available LPA1 receptor antagonist for treating idiopathic pulmonary fibrosis.
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 68 | In Stock |
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| 10MG | 110 | In Stock |
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| 25MG | 200 | In Stock |
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| 50MG | 335 | In Stock |
|
| 100MG | 500 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBMS-986020
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NoteResearch use only, not for human use.
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Brief DescriptionBMS-986020 (BMS986020, AM-152) is a potent, selective, orally available LPA1 receptor antagonist for treating idiopathic pulmonary fibrosis.
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DescriptionBMS-986020 (BMS986020, AM-152) is a potent, selective, orally available LPA1 receptor antagonist for treating idiopathic pulmonary fibrosis.Cystic Fibrosis,Phase 2 Clinical
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SynonymsBMS 986020;BMS986020;AM-152;AM152;AM 152
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PathwayGPCR/G Protein
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TargetLysophospholipid Receptor
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RecptorLPA1
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Research AreaOther Indications
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IndicationFibrosis
Chemical Information
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CAS Number1257213-50-5
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Formula Weight482.53
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Molecular FormulaC29H26N2O5
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Purity>98%(HPLC)
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SolubilityDMSO: ≥ 64 mg/mL
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SMILESCC1=NOC(=C1NC(=O)OC(C)C2=CC=CC=C2)C3=CC=C(C=C3)C4=CC=C(C=C4)C5(CC5)C(=O)O
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Chemical NameCyclopropanecarboxylic acid, 1-[4'-[3-methyl-4-[[[(1R)-1-phenylethoxy]carbonyl]amino]-5-isoxazolyl][1,1'-biphenyl]-4-yl]-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Kihara Y, et al. Exp Cell Res. 2015 May 1;333(2):171-7.
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