BML-210
CAS No. 537034-17-6
BML-210 ( BML210;BML 210 )
Catalog No. M14907 CAS No. 537034-17-6
A novel histone deacetylase (HDAC) inhibitor that induces Ac-histone in A549 cells with EC50 of 181 uM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
2MG | 31 | In Stock |
|
5MG | 48 | In Stock |
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10MG | 69 | In Stock |
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25MG | 115 | In Stock |
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50MG | 186 | In Stock |
|
100MG | 332 | In Stock |
|
200MG | Get Quote | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
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Biological Information
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Product NameBML-210
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NoteResearch use only, not for human use.
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Brief DescriptionA novel histone deacetylase (HDAC) inhibitor that induces Ac-histone in A549 cells with EC50 of 181 uM.
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DescriptionA novel histone deacetylase (HDAC) inhibitor that induces Ac-histone in A549 cells with EC50 of 181 uM; inhibits the growth of all cell lines and promotes apoptosis in the human leukemia cell lines (NB4, HL-60, THP-1, and K562); induces growth inhibition and apoptosis and downregulates HDAC1-5 and DAPC complex expression levels in cervical cancer cells.
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SynonymsBML210;BML 210
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PathwayCell Cycle/DNA Damage
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TargetHDAC
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RecptorHDAC
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number537034-17-6
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Formula Weight339.43
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Molecular FormulaC20H25N3O2
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 30 mg/mL
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SMILESO=C(NC1=CC=CC=C1N)CCCCCCC(NC2=CC=CC=C2)=O
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Chemical NameOctanediamide, N1-(2-aminophenyl)-N8-phenyl-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Savickiene J, et al. Eur J Pharmacol. 2006 Nov 7;549(1-3):9-18.
2. Wong JC, et al. J Am Chem Soc. 2003 May 14;125(19):5586-7.
3. Borutinskaite VV, et al. Mol Biol Rep. 2012 Dec;39(12):10179-86.
2. Wong JC, et al. J Am Chem Soc. 2003 May 14;125(19):5586-7.
3. Borutinskaite VV, et al. Mol Biol Rep. 2012 Dec;39(12):10179-86.
molnova catalog
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