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Home - Products - GPCR/G Protein - Cannabinoid Receptor - WIN 55,212-2 mesylate

WIN 55,212-2 mesylate

CAS No. 131543-23-2

WIN 55,212-2 mesylate( R)-(+)-WIN 55212 | WIN 55212-2 )

Catalog No. M11277 CAS No. 131543-23-2

WIN 55,212-2 mesylate (WIN 55212-2) is a potent cannabinoid receptor agonist with Ki of 62.3 and 3.3 nM for human recombinant CB1 and CB2 receptors, respectively.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    WIN 55,212-2 mesylate
  • Note
    Research use only, not for human use.
  • Brief Description
    WIN 55,212-2 mesylate (WIN 55212-2) is a potent cannabinoid receptor agonist with Ki of 62.3 and 3.3 nM for human recombinant CB1 and CB2 receptors, respectively.
  • Description
    WIN 55,212-2 mesylate (WIN 55212-2) is a potent cannabinoid receptor agonist with Ki of 62.3 and 3.3 nM for human recombinant CB1 and CB2 receptors, respectively; increases extracellular glutamate levels, displaying a bell-shaped concentration-response curve at 0.01-100 nM; increases dialysate glutamate levels the prefrontal cortex from of the awake rats, also demonstrates anticonvulsant effect in vivo pre-treated with 20 mg/kg of pioglitazone.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    R)-(+)-WIN 55212 | WIN 55212-2
  • Pathway
    GPCR/G Protein
  • Target
    Cannabinoid Receptor
  • Recptor
    CB1R|CB2R
  • Research Area
    Neurological Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    131543-23-2
  • Formula Weight
    522.616
  • Molecular Formula
    C28H30N2O6S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: ≥ 34 mg/mL
  • SMILES
    O=C(C1=C(C)N2[C@H](CN3CCOCC3)COC4=CC=CC1=C24)C5=C6C=CC=CC6=CC=C5.CS(=O)(O)=O
  • Chemical Name
    Methanone, [(3R)-2,3-dihydro-5-methyl-3-(4-morpholinylmethyl)pyrrolo[1,2,3-de]-1,4-benzoxazin-6-yl]-1-naphthalenyl-, methanesulfonate (1:1)

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Felder CC, et al. Mol Pharmacol. 1995 Sep;48(3):443-50. 2. Griffin G, et al. J Pharmacol Exp Ther. 1998 May;285(2):553-60. 3. D'Ambra TE, et al. J Med Chem. 1992 Jan;35(1):124-35. 4. Martellotta MC, et al. Neuroscience. 1998 Jul;85(2):327-30.
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