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NESS-040C5
CAS No. 1445751-90-5
NESS-040C5( NESS 040C5 | NESS040C5 )
Catalog No. M11886 CAS No. 1445751-90-5
A potent, reasonably selective cannabinoid CB2 agonist with Ki of 0.4 nM, 25-fold selectivity over CB1 receptor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameNESS-040C5
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NoteResearch use only, not for human use.
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Brief DescriptionA potent, reasonably selective cannabinoid CB2 agonist with Ki of 0.4 nM, 25-fold selectivity over CB1 receptor.
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DescriptionA potent, reasonably selective cannabinoid CB2 agonist with Ki of 0.4 nM, 25-fold selectivity over CB1 receptor.
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In Vitro——
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In Vivo——
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SynonymsNESS 040C5 | NESS040C5
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PathwayGPCR/G Protein
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TargetCannabinoid Receptor
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RecptorCannabinoid Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number1445751-90-5
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Formula Weight447.64
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Molecular FormulaC27H33N3OS
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical NameThieno[3',2':4,5]cyclopenta[1,2-c]pyrazole-3-carboxamide, 1,4-dihydro-N-[5-methyl-2-(1-methylethyl)cyclohexyl]-1-[(4-methylphenyl)methyl]-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Hanus LO, et al. Curr Med Chem. 2010;17(14):1341-59.
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