Cart
sales@molnova.com
NESS-040C5
CAS No. 1445751-90-5
NESS-040C5( NESS 040C5 | NESS040C5 )
Catalog No. M11886 CAS No. 1445751-90-5
A potent, reasonably selective cannabinoid CB2 agonist with Ki of 0.4 nM, 25-fold selectivity over CB1 receptor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 100MG | Get Quote | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameNESS-040C5
-
NoteResearch use only, not for human use.
-
Brief DescriptionA potent, reasonably selective cannabinoid CB2 agonist with Ki of 0.4 nM, 25-fold selectivity over CB1 receptor.
-
DescriptionA potent, reasonably selective cannabinoid CB2 agonist with Ki of 0.4 nM, 25-fold selectivity over CB1 receptor.
-
In Vitro——
-
In Vivo——
-
SynonymsNESS 040C5 | NESS040C5
-
PathwayGPCR/G Protein
-
TargetCannabinoid Receptor
-
RecptorCannabinoid Receptor
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number1445751-90-5
-
Formula Weight447.64
-
Molecular FormulaC27H33N3OS
-
Purity>98% (HPLC)
-
Solubility——
-
SMILES——
-
Chemical NameThieno[3',2':4,5]cyclopenta[1,2-c]pyrazole-3-carboxamide, 1,4-dihydro-N-[5-methyl-2-(1-methylethyl)cyclohexyl]-1-[(4-methylphenyl)methyl]-
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Hanus LO, et al. Curr Med Chem. 2010;17(14):1341-59.
molnova catalog
related products
-
AM-2232
AM-2232 is a potent and unselective agonist of the cannabinoid receptors.
-
AM251
AM251 is a potent CB1 receptor antagonist (IC50 = 8 nM, Ki = 7.49 nM) that displays 306-fold selectivity over CB2 receptors; also potent GPR55 agonist (EC50 = 39 nM).
-
CB2R PAM
CB2R PAM is an orally active cannabinoid type 2 receptor (CB2Rs) positive allosteric modulator that enhances CP 55940 and 2-Arachidonylglycerol-stimulated [35S]GTPγS binding to CB2 receptors without affecting receptor activity in the absence of agonists.
