VUF10460
CAS No. 1028327-66-3
VUF10460( —— )
Catalog No. M17121 CAS No. 1028327-66-3
VUF10460 is a non-imidazole histamine H4 receptor agonist.
Purity : >98% (HPLC)
Size | Price / USD | Stock | Quantity |
2MG | 29 | In Stock |
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5MG | 47 | In Stock |
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10MG | 77 | In Stock |
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25MG | 149 | In Stock |
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50MG | 259 | In Stock |
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100MG | 405 | In Stock |
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200MG | Get Quote | In Stock |
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500MG | Get Quote | In Stock |
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1G | Get Quote | In Stock |
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Biological Information
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Product NameVUF10460
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NoteResearch use only, not for human use.
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Brief DescriptionVUF10460 is a non-imidazole histamine H4 receptor agonist.
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DescriptionVUF10460 is a non-imidazole histamine H4 receptor agonist.
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In VitroUF10460 binds to rat H3 and H4 receptor with pKi values of 5.75, and 7.46, respectively. VUF10460 displays approximately a 50-fold selectivity for the rat H4 receptor over the H3 receptor.
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In VivoHCl-induced rat gastric lesions is significantly enhanced by the H4 receptor agonists VUF10460. This effect is not modified by H4 receptor antagonist JNJ7777120.
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorH4 receptor
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Research AreaInflammation/Immunology
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Indication——
Chemical Information
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CAS Number1028327-66-3
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Formula Weight269.35
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Molecular FormulaC15H19N5
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Purity>98% (HPLC)
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SolubilityDMSO : ≥ 36 mg/mL 133.66 mM
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SMILESCN1CCN(CC1)c1cc(c2ccccc2)nc(N)n1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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12-Dihexadecanoyl-sn...
PE(14:0/14:0) is a phosphatidylethanolamine (PE or GPEtn). It is a glycerophospholipid in which a phosphorylethanolamine moiety occupies a glycerol substitution site. PE(14:0/14:0) in particular consists of two chains of myristic acid at the C-1 and C-2 positions. The myristic acid moieties are derived from nutmeg and butter.
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D-(+)-ALLOSE
D-Allose is a rare naturally occurring monosaccharide known to exert anti-proliferative effects on cancer cells. The effects of D-Allose on the cellular membranes of hormone-refractory prostate cancer cell line (DU145) hormone-sensitive prostate cancer cell line (LNCaP) and normal prostate epithelial cells (PrEC) were studied at the molecular level by phospholipid profiling using a shotgun lipidomic method.
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Adrenocorticotropic ...
Adrenocorticotropic Hormone (ACTH) (1-39), rat is a potent melanocortin 2 (MC2) receptor agonist.Peptide fragments of ACTH (1-39) were formed during in vitro incubation of the peptide with membrane preparations. ACTH (1-39) were isolated by high pressure liquid chromatography, and peptide fragments of ACTH (1-39) characterized by determination of amino acid composition and NH2- terminal residue.