USP8-IN-22e

CAS No. 924296-19-5

USP8-IN-22e ( —— )

Catalog No. M16623 CAS No. 924296-19-5

A potent, selective ubiquitin-specific protease USP8 inhibitor with IC50 of 0.28 uM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 176 Get Quote
5MG 268 Get Quote
10MG 386 Get Quote
25MG 626 Get Quote
50MG 888 Get Quote
100MG 1224 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    USP8-IN-22e
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent, selective ubiquitin-specific protease USP8 inhibitor with IC50 of 0.28 uM.
  • Description
    A potent, selective ubiquitin-specific protease USP8 inhibitor with IC50 of 0.28 uM; shows no inhibitory activity for USP7 (IC50>100 uM).
  • Synonyms
    ——
  • Pathway
    Proteasome/Ubiquitin
  • Target
    DUB
  • Recptor
    DUB
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    924296-19-5
  • Formula Weight
    275.26
  • Molecular Formula
    C15H9N5O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 9.06 mg/mL
  • SMILES
    CCON=C1C2=CC=CC=C2C3=NC(=C(N=C31)C#N)C#N
  • Chemical Name
    9H-Indeno[1,2-b]pyrazine-2,3-dicarbonitrile, 9-(ethoxyimino)-

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Colombo M, et al. ChemMedChem. 2010 Apr 6;5(4):552-8.
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