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UF-010
CAS No. 537672-41-6
UF-010 ( UF010;UF 010 )
Catalog No. M14914 CAS No. 537672-41-6
A potent and selective inhibitor of class I HDACs.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 10MG | 41 | In Stock |
|
| 25MG | 77 | In Stock |
|
| 50MG | 133 | In Stock |
|
| 100MG | 222 | In Stock |
|
| 200MG | 289 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameUF-010
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NoteResearch use only, not for human use.
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Brief DescriptionA potent and selective inhibitor of class I HDACs.
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DescriptionA potent and selective inhibitor of class I HDACs with IC50s of 0.5/0.1/0.06/1.5/9.1/15.3/44.5 uM for HDAC1/2/3/8/6/10/11 respectively; shows no effect on HDAC4/5/7/9(>100 uM); induces the accumulation of protein acetylation and inhibits proliferation of NCI-60 panel of cancer cell lines (mean GI50=2.94 uM); a competitive with a fast-on/slow-off HDAC-binding mechanism.
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SynonymsUF010;UF 010
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PathwayCell Cycle/DNA Damage
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TargetHDAC
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RecptorHDAC
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number537672-41-6
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Formula Weight271.15
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Molecular FormulaC11H15BrN2O
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESO=C(NNCCCC)C1=CC=C(Br)C=C1
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Chemical NameBenzoic acid, 4-bromo-, 2-butylhydrazide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Wang Y, et al. Chem Biol. 2015 Feb 19;22(2):273-84.
molnova catalog
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