TPX-0046

CAS No. 2359650-19-2

TPX-0046 ( —— )

Catalog No. M28037 CAS No. 2359650-19-2

TPX-0046 is a RET inhibitor designed to overcome resistance to Selpercatinib and Pralsetinib.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 209 Get Quote
5MG 335 Get Quote
10MG 520 Get Quote
25MG 1107 Get Quote
50MG 1521 Get Quote
100MG 2052 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    TPX-0046
  • Note
    Research use only, not for human use.
  • Brief Description
    TPX-0046 is a RET inhibitor designed to overcome resistance to Selpercatinib and Pralsetinib.
  • Description
    TPX-0046 is a RET inhibitor designed to overcome resistance to Selpercatinib and Pralsetinib.
  • Synonyms
    ——
  • Pathway
    Proteasome/Ubiquitin
  • Target
    p97
  • Recptor
    BCRP;ABCG2
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2359650-19-2
  • Formula Weight
    424.4
  • Molecular Formula
    C21H21FN6O3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=C1NC[C@@H](C)OC2=NC=C(F)C=C2CN3C4=NC5=C1C=NN5C=C4O[C@@]6([H])[C@]3([H])CCC6
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Milligan SR, et al. The endocrine activities of 8-prenylnaringenin and related hop (Humulus lupulus L.) flavonoids. J Clin Endocrinol Metab. 2000 Dec;85(12):4912-5.
molnova catalog
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