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LC-1028
CAS No. 2324158-08-7
LC-1028( LC1028 | LC 1028 )
Catalog No. M13662 CAS No. 2324158-08-7
LC-1028 (LC1028) is a novel potent selective, covalent and irreversible inhibitor of p97 (valosin-containing protein).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 873 | In Stock |
|
| 50MG | 1782 | In Stock |
|
| 100MG | 2250 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameLC-1028
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NoteResearch use only, not for human use.
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Brief DescriptionLC-1028 (LC1028) is a novel potent selective, covalent and irreversible inhibitor of p97 (valosin-containing protein).
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DescriptionLC-1028 (LC1028) is a novel potent selective, covalent and irreversible inhibitor of p97 (valosin-containing protein), remains essentially irreversible ac tivity against p97 mutant C522A.
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In Vitro——
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In Vivo——
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SynonymsLC1028 | LC 1028
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PathwayProteasome/Ubiquitin
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Targetp97
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Recptorp97
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Research Area——
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Indication——
Chemical Information
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CAS Number2324158-08-7
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Formula Weight449.558
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Molecular FormulaC28H27N5O
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Purity>98% (HPLC)
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Solubility——
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SMILESCC#CC(NC1=CC=CC2=C1C=C(C)N2C3=NC(NCC4=CC=CC=C4)=C5CCCCC5=N3)=O
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Chemical NameN-(1-(4-(Benzylamino)-5,6,7,8-tetrahydroquinazolin-2-yl)-2-methyl-1H-indol-4-yl)but-2-ynamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Ding R, et al. J Med Chem. 2019 Mar 14;62(5):2814-2829.
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