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STD-101-D1
CAS No. 2151041-09-5
STD-101-D1 ( —— )
Catalog No. M13433 CAS No. 2151041-09-5
STD-101-D1 is a novel brain permeable, G protein-biased beta-1 adrenergic receptor (ADRB1) partial agonist with EC50 of 16.9 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameSTD-101-D1
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NoteResearch use only, not for human use.
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Brief DescriptionSTD-101-D1 is a novel brain permeable, G protein-biased beta-1 adrenergic receptor (ADRB1) partial agonist with EC50 of 16.9 nM.
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DescriptionSTD-101-D1 is a novel brain permeable, G protein-biased beta-1 adrenergic receptor (ADRB1) partial agonist with EC50 of 16.9 nM; engages very little beta-arrestin recruitment compared to the unbiased agonist isoproterenol; also inhibits the acute peripheral and CNS TNFα response induced by LPS both in vitro and in vivo.
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Synonyms——
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PathwayAngiogenesis
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TargetAdrenergic Receptor
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RecptorAdrenergic Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number2151041-09-5
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Formula Weight333.38
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Molecular FormulaC18H23NO5
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name(S)-4-(2-hydroxy-3-((2-(2-methoxyphenoxy)ethyl)amino)propoxy)phenol
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Yi B, et al. PLoS One. 2017 Jul 26;12(7):e0180319.
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