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Perospirone

CAS No. 150915-41-6

Perospirone( —— )

Catalog No. M18058 CAS No. 150915-41-6

Perospirone is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors. It also displays affinity towards 5HT1A receptors as a partial agonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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10MG 91 In Stock
25MG 171 In Stock
50MG 309 In Stock
100MG 528 In Stock
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Biological Information

  • Product Name
    Perospirone
  • Note
    Research use only, not for human use.
  • Brief Description
    Perospirone is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors. It also displays affinity towards 5HT1A receptors as a partial agonist.
  • Description
    Perospirone is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors. It also displays affinity towards 5HT1A receptors as a partial agonist.
  • In Vitro
    ——
  • In Vivo
    Animal Model:Male ICR mice (6 weeks old) weighing 25-30 g Dosage:1.0, 3.0 or 10.0 mg/kg Administration:Orally; daily; for 14 consecutive days Result:Significantly attenuated PCP-induced cognitive deficits in mice in a dose-dependent manner.
  • Synonyms
    ——
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    PARP
  • Recptor
    5-HT2A|D2
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    150915-41-6
  • Formula Weight
    426.57
  • Molecular Formula
    C23H30N4O2S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 5 mg/mL (11.72 mM)
  • SMILES
    O=C1[C@H]2CCCC[C@H]2C(=O)N1CCCCN1CCN(CC1)c1nsc2ccccc12
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Ishibashi T, Ohno Y. Perospirone hydrochloride: the novel atypical antipsychotic agent with high affinities for 5-HT2, D2 and 5-HT1A receptors[J]. Biogenic Amines, 2004, 18(3):307-317.
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