Perospirone

CAS No. 150915-41-6

Perospirone( —— )

Catalog No. M18058 CAS No. 150915-41-6

Perospirone is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors. It also displays affinity towards 5HT1A receptors as a partial agonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 55 In Stock
10MG 91 In Stock
25MG 171 In Stock
50MG 309 In Stock
100MG 528 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Perospirone
  • Note
    Research use only, not for human use.
  • Brief Description
    Perospirone is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors. It also displays affinity towards 5HT1A receptors as a partial agonist.
  • Description
    Perospirone is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors. It also displays affinity towards 5HT1A receptors as a partial agonist.
  • In Vitro
    ——
  • In Vivo
    Animal Model:Male ICR mice (6 weeks old) weighing 25-30 g Dosage:1.0, 3.0 or 10.0 mg/kg Administration:Orally; daily; for 14 consecutive days Result:Significantly attenuated PCP-induced cognitive deficits in mice in a dose-dependent manner.
  • Synonyms
    ——
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    PARP
  • Recptor
    5-HT2A|D2
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    150915-41-6
  • Formula Weight
    426.57
  • Molecular Formula
    C23H30N4O2S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 5 mg/mL (11.72 mM)
  • SMILES
    O=C1[C@H]2CCCC[C@H]2C(=O)N1CCCCN1CCN(CC1)c1nsc2ccccc12
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Ishibashi T, Ohno Y. Perospirone hydrochloride: the novel atypical antipsychotic agent with high affinities for 5-HT2, D2 and 5-HT1A receptors[J]. Biogenic Amines, 2004, 18(3):307-317.
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