PPT

CAS No. 263717-53-9

PPT( PPT )

Catalog No. M13809 CAS No. 263717-53-9

An allosteric GABAA receptor modulator that strongly suppresses GABA-induced chloride currents.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 80 In Stock
10MG 129 In Stock
25MG 251 In Stock
50MG 447 In Stock
100MG 669 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
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Biological Information

  • Product Name
    PPT
  • Note
    Research use only, not for human use.
  • Brief Description
    An allosteric GABAA receptor modulator that strongly suppresses GABA-induced chloride currents.
  • Description
    An allosteric GABAA receptor modulator that strongly suppresses GABA-induced chloride currents.
  • In Vitro
    The EC50 of Propyl pyrazole triol for the ERα-dependent response is 140 pM in ERα-U2OS-Luc cells.
  • In Vivo
    ——
  • Synonyms
    PPT
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    GAT
  • Recptor
    GAT
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    263717-53-9
  • Formula Weight
    388.467
  • Molecular Formula
    C24H24N2O3
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : ≥ 100 mg/mL (258.77 mM)
  • SMILES
    OC1=CC=C(C2=C(CCC)C(C3=CC=C(O)C=C3)=NN2C4=CC=C(O)C=C4)C=C1
  • Chemical Name
    4,4',4″-(4-propyl-[1H]-pyrazole-1,3,5-triyl)trisphenol

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Yamaura K, et al. Nat Chem Biol. 2016 Oct;12(10):822-30.
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