MK-0773
CAS No. 606101-58-0
MK-0773 ( MK0773;MK 0773;PF 05314882;PF-05314882;PF05314882 )
Catalog No. M15267 CAS No. 606101-58-0
A potent, selective androgen receptor modulator (SARM) with binding IC50 of 6.6 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
10MG | 417 | Get Quote |
|
50MG | 988 | Get Quote |
|
100MG | Get Quote | Get Quote |
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200MG | Get Quote | Get Quote |
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500MG | Get Quote | Get Quote |
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1G | Get Quote | Get Quote |
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Biological Information
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Product NameMK-0773
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NoteResearch use only, not for human use.
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Brief DescriptionA potent, selective androgen receptor modulator (SARM) with binding IC50 of 6.6 nM.
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DescriptionA potent, selective androgen receptor modulator (SARM) with binding IC50 of 6.6 nM; displays no binding to other nuclear receptors ( GR, IC50> 2 uM) and 5α-reductase (IC50>10 uM); improves muscle function while minimizing effects on other tissues.Osteoporosis Phase 1 Clinical
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SynonymsMK0773;MK 0773;PF 05314882;PF-05314882;PF05314882
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PathwayEndocrinology/Hormones
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TargetAndrogen Receptor (AR)
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RecptorAndrogen Receptor (AR)
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Research AreaMetabolic Disease
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IndicationOsteoporosis
Chemical Information
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CAS Number606101-58-0
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Formula Weight479.59
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Molecular FormulaC27H34FN5O2
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESC[C@@]12[C@@H](C(NCC3=NC4=CC=CN=C4N3)=O)CC[C@@]1([H])[C@]5([H])CC[C@@]6([H])N(C)C(C(F)=C[C@]6(C)[C@@]5([H])CC2)=O
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Chemical Name1H-Indeno[5,4-f]quinoline-7-carboxamide, 3-fluoro-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-N-(3H-imidazo[4,5-b]pyridin-2-ylmethyl)-1,4a,6a-trimethyl-2-oxo-, (4aS,4bS,6aS,7S,9aS,9bS,11aR)-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Schmidt A, et al. J Biol Chem. 2010 May 28;285(22):17054-64.
2. Papanicolaou DA, et al. J Nutr Health Aging. 2013;17(6):533-43.
2. Papanicolaou DA, et al. J Nutr Health Aging. 2013;17(6):533-43.
molnova catalog
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