MS177 is an effective and fast-acting EZH2 degrader. MS177 is a PROTAC that consists of a CRBN ligand, linker, and a potent enzymatic EZH2 inhibitor C24 (C24 IC50): 12?nM). MS177 effectively depletes both canonical EZH2–PRC2 and noncanonical EZH2–cMyc complexes. MS177 induces leukaemia cell growth inhibition, apoptosis and cell cycle progression arrest.

Antennapedia Peptide TFA is a 16 amino acid peptide (RQIKIWFQNRRMKWKK). The DNA binding domain of the Drosophila transcription factor (Antennapedia), a 60 amino acid protein, is rapidly taken up by cells and has been fused to selected antigens to enhance their immunogenicity. A 16 amino acid peptide Antennapedia Peptide TFA from Antennapedia can facilitate the cytoplasmic uptake of cytotoxic T lymphocyte epitope 9-mer peptides.

Camelliaside A is a compound with the anti-inflammatory effect.