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FLT3-IN-16
CAS No. 298207-49-5
FLT3-IN-16( —— )
Catalog No. M37680 CAS No. 298207-49-5
FLT3-IN-16 exhibits potent inhibitory activity against FLT3 tyrosine kinase with an IC 50 of 1.1 μM. FLT3-IN-16 can be used for researching acute myeloid leukemia .
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 53 | In Stock |
|
| 2MG | 29 | In Stock |
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| 5MG | 48 | In Stock |
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| 10MG | 79 | In Stock |
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| 25MG | 181 | In Stock |
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| 50MG | 269 | In Stock |
|
| 100MG | 381 | In Stock |
|
| 200MG | 503 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameFLT3-IN-16
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NoteResearch use only, not for human use.
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Brief DescriptionFLT3-IN-16 exhibits potent inhibitory activity against FLT3 tyrosine kinase with an IC 50 of 1.1 μM. FLT3-IN-16 can be used for researching acute myeloid leukemia .
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DescriptionFLT3-IN-16 is a potent FLT3 inhibitor with an IC50 of 1.1 μM. FLT3-IN-16 can be used for researching acute myeloid leukemia.
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In VitroFLT3-IN-16 (compound 9, 0-10 μM) exhibits anti-proliferative activities against MV4-11 cells with an IC50 value of 2.0 μM.
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorOthers
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Research Area——
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Indication——
Chemical Information
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CAS Number298207-49-5
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Formula Weight301.36
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Molecular FormulaC15H15N3O2S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 25 mg/mL (82.96 mM; Ultrasonic (<80°C)
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SMILESNC(=O)c1c(NC(=O)c2cccnc2)sc2CCCCc12
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Patch RJ, et, al. Identification of 2-acylaminothiophene-3-carboxamides as potent inhibitors of FLT3. Bioorg Med Chem Lett. 2006 Jun 15;16(12):3282-6.?
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