D4R agonist-1
CAS No. 2826198-44-9
D4R agonist-1( —— )
Catalog No. M37215 CAS No. 2826198-44-9
D4R agonist-1 is a selective and potent D4R partial agonist (Ki:2.2 nM).D4R agonist-1 can be used to study neurological diseases.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 645 | In Stock |
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| 10MG | 798 | In Stock |
|
| 25MG | 1055 | In Stock |
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| 100MG | Get Quote | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameD4R agonist-1
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NoteResearch use only, not for human use.
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Brief DescriptionD4R agonist-1 is a selective and potent D4R partial agonist (Ki:2.2 nM).D4R agonist-1 can be used to study neurological diseases.
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DescriptionD4R agonist-1 (Compound 16f) is a D4R partial agonist (Ki: 2.2 nM). D4R agonist-1 is metabolically stable in rat and human liver microsomes. D4R agonist-1 can be used for research of neuropsychiatric disorders.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetDopamine Receptor
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RecptorDopamine Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number2826198-44-9
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Formula Weight338.47
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Molecular FormulaC19H22N4S
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Purity>98% (HPLC)
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Solubility——
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SMILESN=1C=CC=CC1N2CCN(CC2)CCCC3=NC=4C=CC=CC4S3
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Boateng CA, et al. Pharmacology and Therapeutic Potential ofBenzothiazole Analogues for Cocaine Use Disorder. J Med Chem. 2023 Aug 30.?
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