D4R agonist-1

CAS No. 2826198-44-9

D4R agonist-1( —— )

Catalog No. M37215 CAS No. 2826198-44-9

D4R agonist-1 is a selective and potent D4R partial agonist (Ki:2.2 nM).D4R agonist-1 can be used to study neurological diseases.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    D4R agonist-1
  • Note
    Research use only, not for human use.
  • Brief Description
    D4R agonist-1 is a selective and potent D4R partial agonist (Ki:2.2 nM).D4R agonist-1 can be used to study neurological diseases.
  • Description
    D4R agonist-1 (Compound 16f) is a D4R partial agonist (Ki: 2.2 nM). D4R agonist-1 is metabolically stable in rat and human liver microsomes. D4R agonist-1 can be used for research of neuropsychiatric disorders.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Dopamine Receptor
  • Recptor
    Dopamine Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2826198-44-9
  • Formula Weight
    338.47
  • Molecular Formula
    C19H22N4S
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    N=1C=CC=CC1N2CCN(CC2)CCCC3=NC=4C=CC=CC4S3
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Boateng CA, et al. Pharmacology and Therapeutic Potential ofBenzothiazole Analogues for Cocaine Use Disorder. J Med Chem. 2023 Aug 30.?
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