D4R agonist-1

CAS No. 2826198-44-9

D4R agonist-1( —— )

Catalog No. M37215 CAS No. 2826198-44-9

D4R agonist-1 is a selective and potent D4R partial agonist (Ki:2.2 nM).D4R agonist-1 can be used to study neurological diseases.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 532 Get Quote
5MG 922 Get Quote
10MG 1140 Get Quote
25MG 1463 Get Quote
50MG 1822 Get Quote
100MG 2250 Get Quote
500MG 4419 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    D4R agonist-1
  • Note
    Research use only, not for human use.
  • Brief Description
    D4R agonist-1 is a selective and potent D4R partial agonist (Ki:2.2 nM).D4R agonist-1 can be used to study neurological diseases.
  • Description
    D4R agonist-1 (Compound 16f) is a D4R partial agonist (Ki: 2.2 nM). D4R agonist-1 is metabolically stable in rat and human liver microsomes. D4R agonist-1 can be used for research of neuropsychiatric disorders.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Dopamine Receptor
  • Recptor
    Dopamine Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2826198-44-9
  • Formula Weight
    338.47
  • Molecular Formula
    C19H22N4S
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    N=1C=CC=CC1N2CCN(CC2)CCCC3=NC=4C=CC=CC4S3
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Boateng CA, et al. Pharmacology and Therapeutic Potential ofBenzothiazole Analogues for Cocaine Use Disorder. J Med Chem. 2023 Aug 30.?
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