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D4R agonist-1

CAS No. 2826198-44-9

D4R agonist-1( —— )

Catalog No. M37215 CAS No. 2826198-44-9

D4R agonist-1 is a selective and potent D4R partial agonist (Ki:2.2 nM).D4R agonist-1 can be used to study neurological diseases.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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Biological Information

Product Name

D4R agonist-1
Note

Research use only, not for human use.
Brief Description

D4R agonist-1 is a selective and potent D4R partial agonist (Ki:2.2 nM).D4R agonist-1 can be used to study neurological diseases.
Description

D4R agonist-1 (Compound 16f) is a D4R partial agonist (Ki: 2.2 nM). D4R agonist-1 is metabolically stable in rat and human liver microsomes. D4R agonist-1 can be used for research of neuropsychiatric disorders.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

GPCR/G Protein
Target

Dopamine Receptor
Recptor

Dopamine Receptor
Research Area

——
Indication

——

Chemical Information

CAS Number

2826198-44-9
Formula Weight

338.47
Molecular Formula

C19H22N4S
Purity

>98% (HPLC)
Solubility

——
SMILES

N=1C=CC=CC1N2CCN(CC2)CCCC3=NC=4C=CC=CC4S3
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Boateng CA, et al. Pharmacology and Therapeutic Potential ofBenzothiazole Analogues for Cocaine Use Disorder. J Med Chem. 2023 Aug 30.?

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