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CYP1B1-IN-5

CAS No. 176442-56-1

CYP1B1-IN-5( —— )

Catalog No. M36491 CAS No. 176442-56-1

CYP1B1-IN-5 is a selective and potent cytochrome P450 1B1 (CYP1B1) inhibitor with an IC50 of 4.7 nM.CYP1B1-IN-5 can be used for the study of metabolism-related diseases.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
5MG	459	In Stock
10MG	657	In Stock
25MG	1026	In Stock
50MG	1386	In Stock
100MG	1832	In Stock
200MG	Get Quote	In Stock
500MG	3655	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

CYP1B1-IN-5
Note

Research use only, not for human use.
Brief Description

CYP1B1-IN-5 is a selective and potent cytochrome P450 1B1 (CYP1B1) inhibitor with an IC50 of 4.7 nM.CYP1B1-IN-5 can be used for the study of metabolism-related diseases.
Description

CYP1B1-IN-5 (Compound 6q) is a potent and selective cytochrome P450 1B1 (CYP1B1) inhibitor with an IC50 of 4.7 nM.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

Metabolic Enzyme/Protease
Target

P450
Recptor

P450
Research Area

——
Indication

——

Chemical Information

CAS Number

176442-56-1
Formula Weight

349.12
Molecular Formula

C14H8INO2
Purity

>98% (HPLC)
Solubility

——
SMILES

O=C1OC(=NC=2C1=CC=CC2)C3=CC=C(I)C=C3
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Yi L, et al. A new class of CYP1B1 inhibitors derived from bentranil. Bioorg Med Chem Lett. 2022 Dec 21;80:129112.?

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