USP1-IN-2

CAS No. 2098212-05-4

USP1-IN-2( —— )

Catalog No. M35724 CAS No. 2098212-05-4

USP1-IN-2 is a potent USP1 inhibitor with potential anti-tumor activity for the study of cancer.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 445 Get Quote
5MG 686 Get Quote
10MG 905 Get Quote
25MG 1334 Get Quote
50MG 1730 Get Quote
100MG 2313 Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    USP1-IN-2
  • Note
    Research use only, not for human use.
  • Brief Description
    USP1-IN-2 is a potent USP1 inhibitor with potential anti-tumor activity for the study of cancer.
  • Description
    USP1-IN-2 (Compound I-193) is a potent ubiquitin-specific protease 1 (USP1) inhibitor with an IC50 of less than about 50 nM.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Proteasome/Ubiquitin
  • Target
    DUB
  • Recptor
    DUB
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2098212-05-4
  • Formula Weight
    510.486
  • Molecular Formula
    C26H22F4N6O
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 62.5 mg/mL (122.43 mM; Ultrasonic (<60°C)
  • SMILES
    CC(C)c1c(F)cccc1-c1ncc2[nH]c(=O)n(Cc3ccc(cc3)-c3nc(cn3C)C(F)(F)F)c2n1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Alexandre Joseph Buckmelter, et al. Purinones as ubiquitin-specific protease 1 inhibitors. Patent US20170145012A1.
molnova catalog
related products
  • OTUB1/USP8-IN-1

    OTUB1/USP8-IN-1 is a potent OTUB1/USP8 inhibitor with potential anticancer activity, demonstrating IC50 values of 0.17 nM for OTUB1 and 0.28 nM for USP8.

  • USP8-IN-22e

    A potent, selective ubiquitin-specific protease USP8 inhibitor with IC50 of 0.28 uM.

  • NSC112200

    NSC112200 is a chemical inhibitor of the EZH2 deubiquitinase ZRANB1 (at 10 uM), destabilizes EZH2.