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Nesuparib
CAS No. 2055357-64-5
Nesuparib( —— )
Catalog No. M35605 CAS No. 2055357-64-5
Nesuparib (JPI-547/OCN-201) is a potent PARP inhibitor with inhibitory effects on PARP and TNKS1.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 233 | In Stock |
|
| 5MG | 211 | In Stock |
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| 10MG | 337 | In Stock |
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| 25MG | 605 | In Stock |
|
| 50MG | 807 | In Stock |
|
| 100MG | 1097 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameNesuparib
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NoteResearch use only, not for human use.
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Brief DescriptionNesuparib (JPI-547/OCN-201) is a potent PARP inhibitor with inhibitory effects on PARP and TNKS1.
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DescriptionNesuparib is a potent inhibitor of PARP. Nesuparib is useful for the research of neuropathic pain, neurodegenerative disease, and cardiovascular disease (extracted from patent WO2016200101A2).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayWnt/Notch/Hedgehog
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TargetWnt/beta/catenin
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RecptorWnt/beta-catenin | PARP
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Research Area——
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Indication——
Chemical Information
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CAS Number2055357-64-5
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Formula Weight400.48
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Molecular FormulaC23H24N6O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : ≥ 62.5 mg/mL (156.06 mM )
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SMILESO=c1[nH]c2cc(CN3CCN(CC3)c3ccc(cn3)C#N)ccc2c2NCCCc12
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Tricyclic derivative compound, method for preparing same, and pharmaceutical composition comprising same. Patent WO2016200101A2.
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