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Metapramine
CAS No. 21730-16-5
Metapramine( —— )
Catalog No. M35401 CAS No. 21730-16-5
Metapramine (19560 RP) is a novel psychostimulant, an N-methyl-D-aspartate receptor (NMDA) antagonist with antidepressant and anti-injury perception activity that promotes increased levels of acetylcholine in the striatum.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 411 | In Stock |
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| 10MG | 562 | In Stock |
|
| 25MG | 866 | In Stock |
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| 100MG | Get Quote | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameMetapramine
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NoteResearch use only, not for human use.
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Brief DescriptionMetapramine (19560 RP) is a novel psychostimulant, an N-methyl-D-aspartate receptor (NMDA) antagonist with antidepressant and anti-injury perception activity that promotes increased levels of acetylcholine in the striatum.
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DescriptionMetapramine (19560 RP) is an antidepressant agent, belonging to the class of tricyclic compounds. Metapramine inhibits norepinephrine reuptake, without affecting the reuptake of serotonin or dopamine. Metapramine is a low-affinity antagonist of the N-methyl-D-aspartic acid (NMDA) receptor complex channel.
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In Vitro——
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In VivoMetapramine (19560 RP) (0-20 mg/kg; i.p.) shows analgesic effects in mice.Animal Model:Male Swiss albino mice Dosage:0-20 mg/kg Administration:Intraperitoneal injection Result:Increased jump latency, threshold voltage, reduction in writhes, and tail flick latency in a dose-dependent manner.
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Synonyms——
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PathwayMetabolic Enzyme/Protease
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TargetDehydrogenase
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RecptorDehydrogenase
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Research Area——
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Indication——
Chemical Information
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CAS Number21730-16-5
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Formula Weight238.33
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Molecular FormulaC16H18N2
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Purity>98% (HPLC)
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Solubility——
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SMILESC=1C=CC2=C(C1)N(C=3C=CC=CC3C(NC)C2)C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. M Bonierbale, et al. [Metapramine: antidepressant and psycho-stimulant]. Encephale. 1976;2(3):219-23.?
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