SCH-900271

CAS No. 915210-50-3

SCH-900271( —— )

Catalog No. M34706 CAS No. 915210-50-3

SCH-900271 is a potent nicotinic acid receptor for the treatment of dyslipidaemia and is commonly used in the study of mixed hyperlipidaemia and primary hypercholesterolaemia.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 262 In Stock
5MG 276 In Stock
10MG 418 In Stock
25MG 692 In Stock
50MG 918 In Stock
100MG 1293 In Stock
200MG Get Quote In Stock
500MG 2576 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    SCH-900271
  • Note
    Research use only, not for human use.
  • Brief Description
    SCH-900271 is a potent nicotinic acid receptor for the treatment of dyslipidaemia and is commonly used in the study of mixed hyperlipidaemia and primary hypercholesterolaemia.
  • Description
    SCH-900271 is an orally active, potent nicotinic acid receptor (NAR) agonist with an EC50 of 2 nM in the hu-GPR109a assay. SCH-900271 exhibits dose-dependent inhibition of plasma free fatty acid (FFA). SCH-900271 has an improved therapeutic window to flushing.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    AChR
  • Recptor
    AChR
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    915210-50-3
  • Formula Weight
    276.29
  • Molecular Formula
    C14H16N2O4
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    C(CCC1(C)CC1)C=2C3=C(NC(=O)NC3=O)OC(=O)C2
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Anandan Palani, et al. Discovery of SCH 900271, a Potent Nicotinic Acid Receptor Agonist for the Treatment of Dyslipidemia. ACS Med Chem Lett. 2011 Nov 24;3(1):63-8.?
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