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SCH-900271
CAS No. 915210-50-3
SCH-900271( —— )
Catalog No. M34706 CAS No. 915210-50-3
SCH-900271 is a potent nicotinic acid receptor for the treatment of dyslipidaemia and is commonly used in the study of mixed hyperlipidaemia and primary hypercholesterolaemia.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 262 | In Stock |
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| 5MG | 276 | In Stock |
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| 10MG | 418 | In Stock |
|
| 25MG | 692 | In Stock |
|
| 50MG | 918 | In Stock |
|
| 100MG | 1293 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | 2576 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameSCH-900271
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NoteResearch use only, not for human use.
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Brief DescriptionSCH-900271 is a potent nicotinic acid receptor for the treatment of dyslipidaemia and is commonly used in the study of mixed hyperlipidaemia and primary hypercholesterolaemia.
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DescriptionSCH-900271 is an orally active, potent nicotinic acid receptor (NAR) agonist with an EC50 of 2 nM in the hu-GPR109a assay. SCH-900271 exhibits dose-dependent inhibition of plasma free fatty acid (FFA). SCH-900271 has an improved therapeutic window to flushing.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayCell Cycle/DNA Damage
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TargetAChR
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RecptorAChR
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Research Area——
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Indication——
Chemical Information
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CAS Number915210-50-3
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Formula Weight276.29
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Molecular FormulaC14H16N2O4
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Purity>98% (HPLC)
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Solubility——
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SMILESC(CCC1(C)CC1)C=2C3=C(NC(=O)NC3=O)OC(=O)C2
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Anandan Palani, et al. Discovery of SCH 900271, a Potent Nicotinic Acid Receptor Agonist for the Treatment of Dyslipidemia. ACS Med Chem Lett. 2011 Nov 24;3(1):63-8.?
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