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Abt-288
CAS No. 948845-91-8
Abt-288( —— )
Catalog No. M34151 CAS No. 948845-91-8
ABT-288 is a selective and potent H3 antagonist for the treatment of mild to moderate Alzheimer's dementia.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 459 | In Stock |
|
| 10MG | 657 | In Stock |
|
| 25MG | 1026 | In Stock |
|
| 50MG | 1386 | In Stock |
|
| 100MG | 1832 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameAbt-288
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NoteResearch use only, not for human use.
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Brief DescriptionABT-288 is a selective and potent H3 antagonist for the treatment of mild to moderate Alzheimer's dementia.
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DescriptionABT-288 is a competitive, potent and selective histamine H3 receptor (H3R) antagonist. ABT-288 has Ki values of 1.9 and 8.2 nM for human and rat H3Rs, respectively. ABT-288 can be used in cognitive impairment research..
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetHistamine Receptor
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RecptorHistamine Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number948845-91-8
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Formula Weight372.46
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Molecular FormulaC23H24N4O
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Purity>98% (HPLC)
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Solubility——
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SMILESCN1C[C@@]2(N(CC[C@@]2(C1)[H])C3=CC=C(C=C3)C4=CC=C(C=C4)N5C(=O)C=CC=N5)[H]
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Esbenshade TA, et al. Pharmacological properties and procognitive effects of ABT-288, a potent and selective histamine H3 receptor antagonist. J Pharmacol Exp Ther. 2012 Oct;343(1):233-45.?
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