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SCH 221510
CAS No. 322473-89-2
SCH 221510( —— )
Catalog No. M33925 CAS No. 322473-89-2
SCH 221510 is an orally available, selective and potent NOP agonist with an EC50 of 12 nM and a Ki of 0.3 nM.SCH 221510 has anxiolytic activity and can be used to study neurological disorders.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 108 | Get Quote |
|
| 5MG | 163 | Get Quote |
|
| 10MG | 264 | Get Quote |
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| 25MG | 517 | Get Quote |
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| 50MG | 821 | Get Quote |
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| 100MG | 1305 | Get Quote |
|
| 200MG | 1755 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameSCH 221510
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NoteResearch use only, not for human use.
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Brief DescriptionSCH 221510 is an orally available, selective and potent NOP agonist with an EC50 of 12 nM and a Ki of 0.3 nM.SCH 221510 has anxiolytic activity and can be used to study neurological disorders.
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DescriptionSCH 221510 is a potent, orally active and selective NOP (nociceptin opioid receptor) agonist, with an EC50 of 12 nM and Ki of 0.3 nM. SCH 221510 shows an anxiolytic-like effect.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayEndocrinology/Hormones
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TargetOpioid Receptor
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RecptorOpioid Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number322473-89-2
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Formula Weight397.55
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Molecular FormulaC28H31NO
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Purity>98% (HPLC)
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Solubility——
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SMILESC(N1[C@@]2(C[C@@](O)(C[C@]1(CC2)[H])C3=CC=CC=C3)[H])(C4=C(C)C=CC=C4)C5=C(C)C=CC=C5
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Varty GB, et al. The anxiolytic-like effects of the novel, orally active nociceptin opioid receptor agonist 8-[bis(2-methylphenyl)methyl]-3-phenyl-8-azabicyclo[3.2.1]octan-3-ol (SCH 221510). J Pharmacol Exp Ther. 2008 Aug;326(2):672-82.?
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