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Methylnaltrexone bromide
CAS No. 73232-52-7
Methylnaltrexone bromide( MRZ 2663BR | Naltrexone methylbromide )
Catalog No. M15801 CAS No. 73232-52-7
A peripherally-acting μ-opioid antagonist that acts to reverse some of the side effects of opioid drugs such as constipation without affecting analgesia or precipitating withdrawals.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 86 | In Stock |
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| 2MG | 45 | In Stock |
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| 5MG | 73 | In Stock |
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| 10MG | 112 | In Stock |
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| 25MG | 190 | In Stock |
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| 50MG | 266 | In Stock |
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| 100MG | 462 | In Stock |
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| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameMethylnaltrexone bromide
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NoteResearch use only, not for human use.
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Brief DescriptionA peripherally-acting μ-opioid antagonist that acts to reverse some of the side effects of opioid drugs such as constipation without affecting analgesia or precipitating withdrawals.
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DescriptionA peripherally-acting μ-opioid antagonist that acts to reverse some of the side effects of opioid drugs such as constipation without affecting analgesia or precipitating withdrawals.Other Indication Approved.
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In Vitro——
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In Vivo——
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SynonymsMRZ 2663BR | Naltrexone methylbromide
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PathwayEndocrinology/Hormones
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TargetOpioid Receptor
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RecptorOpioid Receptor
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Research AreaOther Indications
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IndicationOther Disease
Chemical Information
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CAS Number73232-52-7
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Formula Weight436.3394
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Molecular FormulaC21H26BrNO4
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 31 mg/mL
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SMILESO=C1[C@@](OC2=C(O)C=CC3=C24)([H])[C@@]54CC[N+](C)(CC6CC6)[C@@](C3)([H])[C@]5(O)CC1.[Br-]
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Chemical NameMorphinanium, 17-(cyclopropylmethyl)-4,5-epoxy-3,14-dihydroxy-17-methyl-6-oxo-, bromide, (5α)-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Yuan CS, et al. Eur J Pharmacol. 1995 Mar 24;276(1-2):107-11.
2. Foss JF, et al. Life Sci. 1996;59(15):PL235-8.
3. Foss JF, et al. J Clin Pharmacol. 1993 Aug;33(8):747-51.
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