Methylnaltrexone bromide

CAS No. 73232-52-7

Methylnaltrexone bromide( MRZ 2663BR | Naltrexone methylbromide )

Catalog No. M15801 CAS No. 73232-52-7

A peripherally-acting μ-opioid antagonist that acts to reverse some of the side effects of opioid drugs such as constipation without affecting analgesia or precipitating withdrawals.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 42 Get Quote
5MG 69 Get Quote
10MG 106 Get Quote
25MG 180 Get Quote
50MG 257 Get Quote
100MG 447 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    Methylnaltrexone bromide
  • Note
    Research use only, not for human use.
  • Brief Description
    A peripherally-acting μ-opioid antagonist that acts to reverse some of the side effects of opioid drugs such as constipation without affecting analgesia or precipitating withdrawals.
  • Description
    A peripherally-acting μ-opioid antagonist that acts to reverse some of the side effects of opioid drugs such as constipation without affecting analgesia or precipitating withdrawals.Other Indication Approved.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    MRZ 2663BR | Naltrexone methylbromide
  • Pathway
    Endocrinology/Hormones
  • Target
    Opioid Receptor
  • Recptor
    Opioid Receptor
  • Research Area
    Other Indications
  • Indication
    Other Disease

Chemical Information

  • CAS Number
    73232-52-7
  • Formula Weight
    436.3394
  • Molecular Formula
    C21H26BrNO4
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: ≥ 31 mg/mL
  • SMILES
    O=C1[C@@](OC2=C(O)C=CC3=C24)([H])[C@@]54CC[N+](C)(CC6CC6)[C@@](C3)([H])[C@]5(O)CC1.[Br-]
  • Chemical Name
    Morphinanium, 17-(cyclopropylmethyl)-4,5-epoxy-3,14-dihydroxy-17-methyl-6-oxo-, bromide, (5α)-

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Yuan CS, et al. Eur J Pharmacol. 1995 Mar 24;276(1-2):107-11. 2. Foss JF, et al. Life Sci. 1996;59(15):PL235-8. 3. Foss JF, et al. J Clin Pharmacol. 1993 Aug;33(8):747-51.
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