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CYN 154806 TFA(183658-72-2 free base)
CAS No. ——
CYN 154806 TFA(183658-72-2 free base)( —— )
Catalog No. M30045 CAS No. ——
CYN 154806 (TFA) is a cyclic octapeptide and an effective selective somatostatin sst2 receptor antagonist. For the recombinant sst2, sst1, sst3, sst4 and sst5 receptors, the pIC50 values are 8.58, 5.41, 6.07, 5.76 and 6.48, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 430 | Get Quote |
|
| 10MG | 620 | Get Quote |
|
| 25MG | 972 | Get Quote |
|
| 50MG | 1332 | Get Quote |
|
| 100MG | 1764 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
Biological Information
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Product NameCYN 154806 TFA(183658-72-2 free base)
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NoteResearch use only, not for human use.
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Brief DescriptionCYN 154806 (TFA) is a cyclic octapeptide and an effective selective somatostatin sst2 receptor antagonist. For the recombinant sst2, sst1, sst3, sst4 and sst5 receptors, the pIC50 values are 8.58, 5.41, 6.07, 5.76 and 6.48, respectively.
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DescriptionCYN 154806 (TFA) is a cyclic octapeptide and an effective selective somatostatin sst2 receptor antagonist. For the recombinant sst2, sst1, sst3, sst4 and sst5 receptors, the pIC50 values are 8.58, 5.41, 6.07, 5.76 and 6.48, respectively.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetSomatostatin Receptor
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RecptorSomatostatin Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number——
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Formula Weight1311.36
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Molecular FormulaC58H69F3N12O16S2
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Purity>98% (HPLC)
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SolubilityH2O : 50 mg/mL (38.13 mM; Need ultrasonic)
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SMILES——
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Chemical NameSequence:Ac-FCYWKTCY-NH2 (Disulfide bridge: Cys2-Cys7)
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
Bass RT, et al. Identification and characterization of novel somatostatin antagonists. Mol Pharmacol. 1996 Oct;50(4):709-15.
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CYN 154806
CYN 154806 is a potent and selective somatostatin sst2 receptor antagonist, The pIC50 values are 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant sst2, sst1, sst3, sst4 and sst5 receptors respectively.
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