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Paltusotine
CAS No. 2172870-89-0
Paltusotine( —— )
Catalog No. M28835 CAS No. 2172870-89-0
Paltusotine is a nonpeptide, small molecule somatostatin type 2 (SST2) receptor agonist with high oral bioavailability. Paltusotine maintains GH and IGF-1 levels in acromegaly patients
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 424 | In Stock |
|
| 10MG | 613 | In Stock |
|
| 25MG | 928 | In Stock |
|
| 50MG | 1228 | In Stock |
|
| 100MG | 1655 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePaltusotine
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NoteResearch use only, not for human use.
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Brief DescriptionPaltusotine is a nonpeptide, small molecule somatostatin type 2 (SST2) receptor agonist with high oral bioavailability. Paltusotine maintains GH and IGF-1 levels in acromegaly patients
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DescriptionPaltusotine is a nonpeptide, small molecule somatostatin type 2 (SST2) receptor agonist with high oral bioavailability. Paltusotine maintains GH and IGF-1 levels in acromegaly patients
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetSomatostatin Receptor
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RecptorCCK
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Research Area——
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Indication——
Chemical Information
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CAS Number2172870-89-0
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Formula Weight456.49
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Molecular FormulaC27H22F2N4O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 10 mg/mL (21.91 mM)
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SMILESNC(CC1)CCN1c(c1cc(-c(cccc2C#N)c2O)ccc1nc1)c1-c1cc(F)cc(F)c1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Scarpignato C, et al. Effect of a new potent CCK antagonist, lorglumide, on caerulein- and bombesin-induced pancreatic secretion and growth in the rat. Br J Pharmacol. 1989 Mar;96(3):661-9.
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