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TRPM8 antagonist 3
CAS No. 2102179-29-1
TRPM8 antagonist 3( —— )
Catalog No. M28848 CAS No. 2102179-29-1
TRPM8 antagonist 3 is a blocker of TRPM8 (IC50 = 11 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 86 | In Stock |
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| 5MG | 78 | In Stock |
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| 10MG | 122 | In Stock |
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| 25MG | 201 | In Stock |
|
| 50MG | 287 | In Stock |
|
| 100MG | 405 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameTRPM8 antagonist 3
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NoteResearch use only, not for human use.
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Brief DescriptionTRPM8 antagonist 3 is a blocker of TRPM8 (IC50 = 11 nM).
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DescriptionTRPM8 antagonist 3 is a blocker of TRPM8 (IC50 = 11 nM).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMembrane Transporter/Ion Channel
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TargetTRP/TRPV Channel
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RecptorD3 receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number2102179-29-1
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Formula Weight292.315
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Molecular FormulaC13H12N2O4S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 25 mg/mL (85.53 mM)
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SMILESO=C(C1=C(O)N=C(C2=CC=CC=C2O)S1)N3OCCC3
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Grundt P, et al. Novel heterocyclic trans olefin analogues of N-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl}arylcarboxamides as selective probes with high affinity for the dopamine D3 receptor. J Med Chem. 2005 Feb 10;48(3):839-48.
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