TRPM8 antagonist 3

CAS No. 2102179-29-1

TRPM8 antagonist 3( —— )

Catalog No. M28848 CAS No. 2102179-29-1

TRPM8 antagonist 3 is a blocker of TRPM8 (IC50 = 11 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 86 In Stock
5MG 78 In Stock
10MG 122 In Stock
25MG 201 In Stock
50MG 287 In Stock
100MG 405 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    TRPM8 antagonist 3
  • Note
    Research use only, not for human use.
  • Brief Description
    TRPM8 antagonist 3 is a blocker of TRPM8 (IC50 = 11 nM).
  • Description
    TRPM8 antagonist 3 is a blocker of TRPM8 (IC50 = 11 nM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    TRP/TRPV Channel
  • Recptor
    D3 receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2102179-29-1
  • Formula Weight
    292.315
  • Molecular Formula
    C13H12N2O4S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 25 mg/mL (85.53 mM)
  • SMILES
    O=C(C1=C(O)N=C(C2=CC=CC=C2O)S1)N3OCCC3
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Grundt P, et al. Novel heterocyclic trans olefin analogues of N-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl}arylcarboxamides as selective probes with high affinity for the dopamine D3 receptor. J Med Chem. 2005 Feb 10;48(3):839-48.
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