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TRPM8 antagonist 3

CAS No. 2102179-29-1

TRPM8 antagonist 3( —— )

Catalog No. M28848 CAS No. 2102179-29-1

TRPM8 antagonist 3 is a blocker of TRPM8 (IC50 = 11 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 86 In Stock
5MG 78 In Stock
10MG 122 In Stock
25MG 201 In Stock
50MG 287 In Stock
100MG 405 In Stock
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Biological Information

  • Product Name
    TRPM8 antagonist 3
  • Note
    Research use only, not for human use.
  • Brief Description
    TRPM8 antagonist 3 is a blocker of TRPM8 (IC50 = 11 nM).
  • Description
    TRPM8 antagonist 3 is a blocker of TRPM8 (IC50 = 11 nM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    TRP/TRPV Channel
  • Recptor
    D3 receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2102179-29-1
  • Formula Weight
    292.315
  • Molecular Formula
    C13H12N2O4S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 25 mg/mL (85.53 mM)
  • SMILES
    O=C(C1=C(O)N=C(C2=CC=CC=C2O)S1)N3OCCC3
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Grundt P, et al. Novel heterocyclic trans olefin analogues of N-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl}arylcarboxamides as selective probes with high affinity for the dopamine D3 receptor. J Med Chem. 2005 Feb 10;48(3):839-48.
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