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VX-150
CAS No. 1793080-72-4
VX-150( —— )
Catalog No. M28830 CAS No. 1793080-72-4
VX-150 is a highly selective NaV1.8 inhibitor relative to the other sodium channel subtypes (>400-fold).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 222 | Get Quote |
|
| 10MG | 356 | Get Quote |
|
| 25MG | 599 | Get Quote |
|
| 50MG | 852 | Get Quote |
|
| 100MG | 1152 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameVX-150
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NoteResearch use only, not for human use.
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Brief DescriptionVX-150 is a highly selective NaV1.8 inhibitor relative to the other sodium channel subtypes (>400-fold).
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DescriptionVX-150 is a highly selective NaV1.8 inhibitor relative to the other sodium channel subtypes (>400-fold).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMembrane Transporter/Ion Channel
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TargetSodium Channel
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RecptorFatty Acid Synthase (FASN)
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Research Area——
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Indication——
Chemical Information
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CAS Number1793080-72-4
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Formula Weight516.34
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Molecular FormulaC21H17F4N2O7P
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 125 mg/mL (242.09 mM)
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SMILESCc(cc(cc1)F)c1Oc(cc(C(F)(F)F)cc1)c1C(NC(C=CN1COP(O)(O)=O)=CC1=O)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Rae C, et al. Inhibition of Fatty Acid Synthase Sensitizes Prostate Cancer Cells to Radiotherapy. Radiat Res. 2015 Nov;184(5):482-93.
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