VX-150

CAS No. 1793080-72-4

VX-150( —— )

Catalog No. M28830 CAS No. 1793080-72-4

VX-150 is a highly selective NaV1.8 inhibitor relative to the other sodium channel subtypes (>400-fold).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 159 In Stock
5MG 140 In Stock
10MG 235 In Stock
25MG 471 In Stock
50MG 739 In Stock
100MG 1181 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    VX-150
  • Note
    Research use only, not for human use.
  • Brief Description
    VX-150 is a highly selective NaV1.8 inhibitor relative to the other sodium channel subtypes (>400-fold).
  • Description
    VX-150 is a highly selective NaV1.8 inhibitor relative to the other sodium channel subtypes (>400-fold).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    Sodium Channel
  • Recptor
    Fatty Acid Synthase (FASN)
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1793080-72-4
  • Formula Weight
    516.34
  • Molecular Formula
    C21H17F4N2O7P
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 125 mg/mL (242.09 mM)
  • SMILES
    Cc(cc(cc1)F)c1Oc(cc(C(F)(F)F)cc1)c1C(NC(C=CN1COP(O)(O)=O)=CC1=O)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Rae C, et al. Inhibition of Fatty Acid Synthase Sensitizes Prostate Cancer Cells to Radiotherapy. Radiat Res. 2015 Nov;184(5):482-93.
molnova catalog
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