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BMS-986122

CAS No. 313669-88-4

BMS-986122( BMS 986122 | BMS986122 )

Catalog No. M27859 CAS No. 313669-88-4

BMS 986122 is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1 human osteosarcoma cells expressing μ-opioid receptors (EC50 = 3 μM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 92 In Stock
5MG 92 In Stock
10MG 155 In Stock
25MG 312 In Stock
50MG 461 In Stock
100MG 644 In Stock
200MG 910 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock
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Biological Information

  • Product Name
    BMS-986122
  • Note
    Research use only, not for human use.
  • Brief Description
    BMS 986122 is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1 human osteosarcoma cells expressing μ-opioid receptors (EC50 = 3 μM).
  • Description
    BMS 986122 is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1 human osteosarcoma cells expressing μ-opioid receptors (EC50 = 3 μM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    BMS 986122 | BMS986122
  • Pathway
    Endocrinology/Hormones
  • Target
    Opioid Receptor
  • Recptor
    FAP
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    313669-88-4
  • Formula Weight
    448.77
  • Molecular Formula
    C16H15BrClNO3S2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (222.83 mM)
  • SMILES
    COc1ccc(cc1Br)C1SCCN1S(=O)(=O)c1ccc(Cl)cc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Hui Jin Jung, et al. Identification of BR102910 as a selective fibroblast activation protein (FAP) inhibitor. Bioorg Med Chem Lett. 2021 Apr 1;37:127846.
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