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Adrenorphin(3TFA)
CAS No. 88377-68-8
Adrenorphin(3TFA)( Metorphamide )
Catalog No. M21026 CAS No. 88377-68-8
Adrenorphin(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 230 | Get Quote |
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| 10MG | 346 | Get Quote |
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| 25MG | 622 | Get Quote |
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| 50MG | 933 | Get Quote |
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| 100MG | Get Quote | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameAdrenorphin(3TFA)
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NoteResearch use only, not for human use.
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Brief DescriptionAdrenorphin(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
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DescriptionAdrenorphin(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
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In VitroAdrenorphin (Metorphamide) is a opioid octapeptide from bovine brain, acts as a potent agonist of μ-opioid receptor, with Ki of 12 nM. The binding ratios of Ki for μ-opioid receptor/Ki for δ-opioid receptor of 0.04 and of Ki for μ-opioid receptor/Ki for κ-opioid receptor of 0.46. Adrenorphin potently inhibits catecholamine secretion evoked by 10 μM nicotine in cultured human pheochromocytoma 6 cells, with an IC50 of 1.1 μM.
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In Vivo——
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SynonymsMetorphamide
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PathwayEndocrinology/Hormones
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TargetOpioid Receptor
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Recptorμ-opioid receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number88377-68-8
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Formula Weight984.18
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Molecular FormulaC44H69N15O9S
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Purity>98% (HPLC)
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SolubilityDMSO:50 mg/mL (50.80 mM)
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SMILESCSCCC(NC(=O)C(Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)C(N)Cc1ccc(O)cc1)C(=O)NC(CCCNC(=N)N)C(=O)NC(CCCNC(=N)N)C(=O)NC(C(N)=O)C(C)C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Miyata A Mizuno K Minamino N et al. Regional distribution of adrenorphin in rat brain: Comparative study with PH-8P[J]. Biochemical and Biophysical Research Communications 1984 120(3):1030-1036.
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