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VU 0255035
CAS No. 1135243-19-4
VU 0255035( VU 255035 )
Catalog No. M27733 CAS No. 1135243-19-4
VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 72 | In Stock |
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| 5MG | 65 | In Stock |
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| 10MG | 107 | In Stock |
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| 25MG | 235 | In Stock |
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| 50MG | 352 | In Stock |
|
| 100MG | 523 | In Stock |
|
| 200MG | 728 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameVU 0255035
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NoteResearch use only, not for human use.
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Brief DescriptionVU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM.
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DescriptionVU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM. It reduces pilocarpine-induced seizures in mice. It is used to examine the role of the M1 receptor in diverse situations.
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In Vitro——
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In Vivo——
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SynonymsVU 255035
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PathwayCell Cycle/DNA Damage
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TargetAChR
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number1135243-19-4
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Formula Weight432.52
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Molecular FormulaC18H20N6O3S2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 62.5 mg/mL (144.50 mM)
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SMILESO=C(CCNS(=O)(=O)c1cccc2nsnc12)N1CCN(CC1)c1ccncc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Yang YJ, et al. Effective Killing of Cancer Cells Through ROS-Mediated Mechanisms by AMRI-59 Targeting Peroxiredoxin I. Antioxid Redox Signal. 2016 Mar 10;24(8):453-69.
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