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Home - Products - Cell Cycle/DNA Damage - AChR - VU 0255035

VU 0255035

CAS No. 1135243-19-4

VU 0255035( VU 255035 )

Catalog No. M27733 CAS No. 1135243-19-4

VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 72 In Stock
5MG 65 In Stock
10MG 107 In Stock
25MG 235 In Stock
50MG 352 In Stock
100MG 523 In Stock
200MG 728 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock
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Biological Information

  • Product Name
    VU 0255035
  • Note
    Research use only, not for human use.
  • Brief Description
    VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM.
  • Description
    VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM. It reduces pilocarpine-induced seizures in mice. It is used to examine the role of the M1 receptor in diverse situations.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    VU 255035
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    AChR
  • Recptor
    ——
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1135243-19-4
  • Formula Weight
    432.52
  • Molecular Formula
    C18H20N6O3S2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 62.5 mg/mL (144.50 mM)
  • SMILES
    O=C(CCNS(=O)(=O)c1cccc2nsnc12)N1CCN(CC1)c1ccncc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Yang YJ, et al. Effective Killing of Cancer Cells Through ROS-Mediated Mechanisms by AMRI-59 Targeting Peroxiredoxin I. Antioxid Redox Signal. 2016 Mar 10;24(8):453-69.
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