Cart
sales@molnova.com
Home - Products - GPCR/G Protein - Dopamine Receptor - LE 300

LE 300

CAS No. 274694-98-3

LE 300( —— )

Catalog No. M27648 CAS No. 274694-98-3

LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 208 In Stock
10MG 310 In Stock
25MG 519 In Stock
50MG 724 In Stock
100MG 986 In Stock
200MG Get Quote In Stock
500MG 1972 In Stock
1G Get Quote In Stock
Get Quotation Bulk Inquiry Add to Cart

Biological Information

  • Product Name
    LE 300
  • Note
    Research use only, not for human use.
  • Brief Description
    LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.
  • Description
    LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.(In Vitro):The Kis of LE 300 are 1.9 nM and 7.5 nM in CHO cell membranes expressing human dopamine D1 and D5 receptors, respectively. In a rat tail artery experiment, the pA2 value of LE 300 at the 5-HT2A receptor was 8.32.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Dopamine Receptor
  • Recptor
    FAAH
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    274694-98-3
  • Formula Weight
    290.41
  • Molecular Formula
    C20H22N2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CN1CCc2c(Cc3ccccc3CC1)[nH]c1ccccc21
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Pea F, Cojutti PG, Baraldo M. A 10-Year Experience of Therapeutic Drug Monitoring (TDM) of Linezolid in a Hospital-wide Population of Patients Receiving Conventional Dosing: Is there Enough Evidence for Suggesting TDM in the Majority of Patients? Basic Clin Pharmacol Toxicol. 2017 Apr 17.
Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog
related products

  • BP-897

    BP-897 is the first, potent, selective partial dopamine D3 receptor agonist with Ki of 0.92 nM.

  • Ropinirole hydrochlo...

    Ropinirole a selective dopamine D2 receptors agonist with Ki of 29 nM.

  • Phenelzine

    Phenelzine is an antidepressant and mania drug, which is a monoamine oxidase inhibitor. Its antidepressant effect is similar to that of niacinamide.

Sign In Join Free