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LE 300
CAS No. 274694-98-3
LE 300( —— )
Catalog No. M27648 CAS No. 274694-98-3
LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 208 | In Stock |
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| 10MG | 310 | In Stock |
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| 25MG | 519 | In Stock |
|
| 50MG | 724 | In Stock |
|
| 100MG | 986 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | 1972 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameLE 300
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NoteResearch use only, not for human use.
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Brief DescriptionLE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.
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DescriptionLE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.(In Vitro):The Kis of LE 300 are 1.9 nM and 7.5 nM in CHO cell membranes expressing human dopamine D1 and D5 receptors, respectively. In a rat tail artery experiment, the pA2 value of LE 300 at the 5-HT2A receptor was 8.32.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetDopamine Receptor
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RecptorFAAH
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Research Area——
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Indication——
Chemical Information
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CAS Number274694-98-3
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Formula Weight290.41
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Molecular FormulaC20H22N2
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Purity>98% (HPLC)
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Solubility——
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SMILESCN1CCc2c(Cc3ccccc3CC1)[nH]c1ccccc21
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Pea F, Cojutti PG, Baraldo M. A 10-Year Experience of Therapeutic Drug Monitoring (TDM) of Linezolid in a Hospital-wide Population of Patients Receiving Conventional Dosing: Is there Enough Evidence for Suggesting TDM in the Majority of Patients? Basic Clin Pharmacol Toxicol. 2017 Apr 17.
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