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JNJ-37822681
CAS No. 935776-74-2
JNJ-37822681( JNJ 37822681 | JNJ37822681 )
Catalog No. M27891 CAS No. 935776-74-2
JNJ-37822681 is a novel, highly selective dopamine D receptor antagonist characterized by a rapid dissociation rate from the dopamine D receptor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 201 | In Stock |
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| 2MG | 120 | In Stock |
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| 5MG | 187 | In Stock |
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| 10MG | 283 | In Stock |
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| 25MG | 463 | In Stock |
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| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameJNJ-37822681
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NoteResearch use only, not for human use.
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Brief DescriptionJNJ-37822681 is a novel, highly selective dopamine D receptor antagonist characterized by a rapid dissociation rate from the dopamine D receptor.
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DescriptionJNJ-37822681 is a novel, highly selective dopamine D receptor antagonist characterized by a rapid dissociation rate from the dopamine D receptor.(In Vivo):JNJ-37822681 occupied D2 receptors in rat brain at relatively low doses (ED50 = 0.39 mg/kg) and was effective in animal models of psychosis (e.g., inhibition of apomorphine-induced stereotypy or D-amphetamine/phencyclidine-induced hyperlocomotion).
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In Vitro——
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In Vivo——
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SynonymsJNJ 37822681 | JNJ37822681
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PathwayGPCR/G Protein
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TargetDopamine Receptor
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number935776-74-2
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Formula Weight372.343
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Molecular FormulaC17H17F5N4
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Purity>98% (HPLC)
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Solubility——
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SMILESFc1ccc(CN2CCC(CC2)Nc2ccc(nn2)C(F)(F)F)cc1F
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Zhihui Xiao, et al. A new flavanone glucoside from Abrus precatorius.Chemistry of Natural Compounds volume 48, pages 565-567 (2012).
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