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Home - Products - Membrane Transporter/Ion Channel - Monocarboxylate Transporter - AR-C155858

AR-C155858

CAS No. 496791-37-8

AR-C155858( —— )

Catalog No. M26608 CAS No. 496791-37-8

AR-C155858 is an inhibitor of monocarboxylate transporter MCT1 and MCT2 (Kis: 2.3 nM and 10 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 296 In Stock
5MG 282 In Stock
10MG 491 In Stock
25MG 801 In Stock
50MG 1079 In Stock
100MG 1460 In Stock
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Biological Information

  • Product Name
    AR-C155858
  • Note
    Research use only, not for human use.
  • Brief Description
    AR-C155858 is an inhibitor of monocarboxylate transporter MCT1 and MCT2 (Kis: 2.3 nM and 10 nM).
  • Description
    AR-C155858 is an inhibitor of monocarboxylate transporter MCT1 and MCT2 (Kis: 2.3 nM and 10 nM).(In Vitro):AR-C155858 (10 nM-100 nM) inhibits MCT1/MCT2 C-terminal chimaeras. AR-C155858 inhibits MCT1 expressed in Xenopus oocytes in a time- and concentration-dependent manner. AR-C155858 inhibits MCT2, and the 70% inhibition seen at 10 nM is followed by a gradually increasing inhibition which can only be explained by a Ki value of significantly less than 10 nM.
  • In Vitro
    AR-C155858 (10 nM-100 nM) inhibits MCT1/MCT2 C-terminal chimaeras. AR-C155858 inhibits MCT2, and the 70% inhibition seen at 10 nM is followed by a gradually increasing inhibition which can only be explained by a Ki value of significantly less than 10 nM. AR-C155858 inhibits MCT1 expressed in Xenopus oocytes in a time- and concentration-dependent manner.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    Monocarboxylate Transporter
  • Recptor
    Apoptosis| VD/VDR
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    496791-37-8
  • Formula Weight
    461.54
  • Molecular Formula
    C21H27N5O5S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 70 mg/mL (151.67 mM)
  • SMILES
    CC(C)Cn1c2sc(Cc3c(C)n[nH]c3C)c(C(=O)N3C[C@H](O)CO3)c2c(=O)n(C)c1=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Ryoko Okamoto, et al. Inecalcitol, an analog of 1α,25(OH)(2) D(3) , induces growth arrest of androgen-dependent prostate cancer cells. Int J Cancer. 2012 May 15;130(10):2464-73.
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