Cart
sales@molnova.com
Sigma-1 receptor antagonist 3
CAS No. 1639220-17-9
Sigma-1 receptor antagonist 3( —— )
Catalog No. M26445 CAS No. 1639220-17-9
Sigma-1 receptor antagonist 3 is a more potent and selective antagonist of Sigma-1 (σ1) receptor (Ki = 1.14 nM) than σ2 receptor(Ki = 1239 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 187 | In Stock |
|
| 10MG | 306 | In Stock |
|
| 25MG | 503 | In Stock |
|
| 50MG | 668 | In Stock |
|
| 100MG | 886 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameSigma-1 receptor antagonist 3
-
NoteResearch use only, not for human use.
-
Brief DescriptionSigma-1 receptor antagonist 3 is a more potent and selective antagonist of Sigma-1 (σ1) receptor (Ki = 1.14 nM) than σ2 receptor(Ki = 1239 nM).
-
DescriptionSigma-1 receptor antagonist 3 is a more potent and selective antagonist of Sigma-1 (σ1) receptor (Ki = 1.14 nM) than σ2 receptor(Ki = 1239 nM). Sigma-1 receptor antagonist 3 inhibits Human Ether-a-go-go-Related Gene (hERG, IC50 = 1.54 μM).
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayAutophagy
-
TargetSigma receptor
-
Recptor——
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number1639220-17-9
-
Formula Weight363.86
-
Molecular FormulaC19H23ClFN3O
-
Purity>98% (HPLC)
-
SolubilityIn Vitro:?DMSO : 12.5 mg/mL (34.35 mM)
-
SMILESCc1nc(nc(OCCCN2CCCCC2)c1Cl)-c1ccc(F)cc1
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Diaz G, et al. Mitochondrial localization of reactive oxygen species by dihydrofluorescein probes. Histochem Cell Biol. 2003 Oct;120(4):319-25.
molnova catalog
related products
-
Sigma-1 receptor ant...
Sigma-1 receptor antagonist 2 is a more potent and selective antagonist of sigma 1 receptor (σ1 R, Ki = 3.88 nM) than σ2 receptor (Ki = 1288 nM).
-
BD1047.2HBr
BD-1047 dihydrobromide is a selective functional antagonist of sigma receptors.
-
PRE-084 hydrochlorid...
PRE-084 hydrochloride is a selective agonist of σ1(IC50:44 nM, in the sigma receptor assay).
